SCHEMBL6602387

SCHEMBL6602387

CCCN(CCC)CCOc1cc(NC(=O)c2ccco2)ccc1OC

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.59
SMN1; SMN2 Q16637 6/20 0.58
RAB9A P51151 3/20 0.58
TP53 P04637 3/20 0.58
KDM4E B2RXH2 3/20 0.58
NPC1 O15118 2/20 0.58
ESR1 P03372 1/20 0.58
ESR2 Q92731 1/20 0.58
MAPT P10636 8/20 0.56
ALDH1A1 P00352 4/20 0.56
KMT2A Q03164 3/20 0.56
MEN1 O00255 2/20 0.56
HPGD P15428 3/20 0.52
HSD17B10 Q99714 2/20 0.52
HTT P42858 1/20 0.52
LMNA P02545 1/20 0.52
MAPK1 P28482 1/20 0.52
POLB P06746 1/20 0.52
MCHR1 Q99705 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6608917 0.93 TSHR (0.60) TSHRSMN1; SMN2RAB9ATP53KDM4E
SCHEMBL6602432 0.89 TSHR (0.63) TSHRSMN1; SMN2RAB9ATP53KDM4E
SCHEMBL6602378 0.86 MCHR1 (0.64) TSHRSMN1; SMN2RAB9ATP53KDM4E
SCHEMBL6899096 0.82 MCHR1 (0.70) MCHR1
SCHEMBL7614829 0.82 MAPT (0.55) SMN1; SMN2RAB9ATP53KDM4ENPC1
SCHEMBL6604033 0.80 KMT2A (0.55) SMN1; SMN2RAB9AKDM4ENPC1MAPT
SCHEMBL6898088 0.80 MCHR1 (0.67) SMN1; SMN2RAB9ATP53NPC1ALDH1A1
SCHEMBL6921907 0.80 MCHR1 (0.80) MCHR1
SCHEMBL6896989 0.80 MCHR1 (0.67) SMN1; SMN2RAB9ATP53NPC1ALDH1A1
SCHEMBL6605524 0.80 KMT2A (0.68) TSHRSMN1; SMN2RAB9ATP53KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1102535-A4 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORP (US) 2004-09-29 EP disclosed
EP-1102535-A2 COMPOUNDS AND METHODS SmithKline Beecham Corporation (US) 2001-05-30 EP disclosed
WO-2000006085-A2 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2000-02-10 WO disclosed