SCHEMBL6602790

SCHEMBL6602790

COC(=O)CCN1CCN(CC2CN(c3ccc(C(=N)NC(=O)C(c4ccccc4)c4ccccc4)cc3)C(=O)O2)CC1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 3/20 0.48
ITGA2B P08514 3/20 0.48
SIGMAR1 Q99720 13/20 0.45
GRM2 Q14416 1/20 0.40
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
HTR2B P41595 2/20 0.38
F10 P00742 2/20 0.37
PRSS1 P07477 2/20 0.37
PRSS2 P07478 2/20 0.37
PRSS3 P35030 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6605091 0.93 ITGB3 (0.44) ITGB3ITGA2BSIGMAR1GRM2HTR2B
SCHEMBL6600339 0.93 ITGB3 (0.53) ITGB3ITGA2BSIGMAR1GRM2ALDH1A1
SCHEMBL6601630 0.93 ITGB3 (0.53) ITGB3ITGA2BSIGMAR1GRM2HTR2B
SCHEMBL6601247 0.92 ITGB3 (0.44) ITGB3ITGA2BSIGMAR1GRM2HTR2B
SCHEMBL7313131 0.92 ITGB3 (0.43) ITGB3ITGA2BSIGMAR1GRM2HTR2B
SCHEMBL6606277 0.91 ITGB3 (0.44) ITGB3ITGA2BSIGMAR1GRM2F10
SCHEMBL6603429 0.90 ITGB3 (0.46) ITGB3ITGA2BSIGMAR1GRM2F10
SCHEMBL6599465 0.89 ITGB3 (0.51) ITGB3ITGA2BSIGMAR1GRM2PRSS1
SCHEMBL6605472 0.89 SIGMAR1 (0.48) ITGB3ITGA2BSIGMAR1GRM2KDM4E
SCHEMBL6600250 0.89 ITGB3 (0.48) ITGB3ITGA2BSIGMAR1GRM2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0741133-B1 Adhesion receptor antagonists MERCK PATENT GMBH (DE) 2004-01-28 EP disclosed
EP-0741133-A2 Adhesion receptor antagonists MERCK PATENT GmbH (DE) 1996-11-06 EP disclosed