SCHEMBL6602876

SCHEMBL6602876

CCCCOC(=O)NC(O)(CCc1cccc(F)c1)C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.41
RAB9A P51151 3/20 0.40
HPGD P15428 2/20 0.40
LMNA P02545 1/20 0.40
ALDH1A1 P00352 1/20 0.39
CYP3A4 P08684 1/20 0.39
TSHR P16473 1/20 0.39
MAPK1 P28482 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
GAA P10253 2/20 0.39
HCAR2 Q8TDS4 1/20 0.39
PPARG P37231 1/20 0.38
PPARA Q07869 1/20 0.38
GLS O94925 1/20 0.38
TAAR1 Q96RJ0 1/20 0.38
CTSK P43235 2/20 0.38
ALOX5 P09917 1/20 0.38
NPC1 O15118 1/20 0.38
CYP1A2 P05177 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6244118 0.90 MEN1 (0.41) POLBRAB9AHPGDLMNAALDH1A1
SCHEMBL5699570 0.87 GAA (0.49) POLBRAB9ALMNAALDH1A1CYP3A4
SCHEMBL6245825 0.82 CTSS (0.51) POLBHPGDLMNAALDH1A1TSHR
SCHEMBL290981 0.78 TDP1 (0.50) POLBRAB9AHPGDLMNAALDH1A1
Water SCHEMBL2946569 0.77 TDP1 (0.49) POLBRAB9AHPGDLMNAALDH1A1
SCHEMBL5774552 0.75 EPHX1 (0.43) POLBALDH1A1HCAR2CYP1A2CYP2C19
SCHEMBL5085119 0.74 CTSK (0.50) PPARGPPARACTSKCTSS
SCHEMBL6261928 0.72 CTSS (0.45) POLBHPGDLMNAALDH1A1TSHR
SCHEMBL6241020 0.72 CTSS (0.45) POLBHPGDLMNAALDH1A1TSHR
SCHEMBL8442388 0.72 KMT2A (0.53) POLBRAB9ALMNAALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1409466-A2 HIV PROTEASE INHIBITORS, COMPOSITIONS CONTAINING THE SAME, THEIR PHARMACEUTICAL USES AND MATERIALS FOR THEIR SYNTHESIS AGOURON PHARMACEUTICALS, INC. (US) 2004-04-21 EP disclosed
WO-2002100844-A2 HIV PROTEASE INHIBITORS, COMPOSITIONS CONTAINING THE SAME, THEIR PHARMACEUTICAL USES AND MATERIALS FOR THEIR SYNTHESIS AGOURON PHARMACEUTICALS, INC. (US) 2002-12-19 WO disclosed