SCHEMBL6602906

SCHEMBL6602906

CC(=O)Nc1nc(-c2cc(C)cc(C)c2)c(-c2c[c]ncc2)s1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 8/20 0.52
ADORA1 P30542 6/20 0.52
ADORA2A P29274 4/20 0.52
ADORA2B P29275 2/20 0.52
CHRM5 P08912 1/20 0.52
HTR2A P28223 1/20 0.52
HTR2C P28335 1/20 0.52
ALDH1A1 P00352 2/20 0.49
MAPT P10636 2/20 0.49
KDM4E B2RXH2 1/20 0.49
LMNA P02545 1/20 0.49
GAA P10253 1/20 0.49
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
DRD4 P21917 1/20 0.46
TSPO P30536 1/20 0.46
DRD3 P35462 1/20 0.46
TMEM97 Q5BJF2 1/20 0.46
PIK3CG P48736 3/20 0.42
PIK3CD O00329 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6545438 0.84 ADORA3 (0.63) ADORA3ADORA1ADORA2AADORA2BCHRM5
SCHEMBL6283239 0.84 ADORA3 (0.69) ADORA3ADORA1ADORA2AADORA2BCHRM5
SCHEMBL3891946 0.82 ALDH1A1 (0.53) ADORA3ADORA1ADORA2AADORA2BCHRM5
SCHEMBL3896156 0.81 ADORA3 (0.54) ADORA3ADORA1ADORA2AADORA2BCHRM5
SCHEMBL3902975 0.81 ADORA3 (0.53) ADORA3ADORA1ADORA2AADORA2BCHRM5
SCHEMBL6545803 0.78 ADORA3 (0.67) ADORA3ADORA1ADORA2AADORA2BCHRM5
SCHEMBL3887415 0.77 ADORA3 (0.52) ADORA3ADORA1ADORA2AADORA2BCHRM5
SCHEMBL6545521 0.77 ALDH1A1 (0.54) ADORA3ADORA1ADORA2AADORA2BCHRM5
SCHEMBL3071322 0.74 ADORA3 (0.62) ADORA3ADORA1ADORA2AADORA2BCHRM5
SCHEMBL4261794 0.74 MAPK14 (0.67) ADORA3ADORA1ADORA2AADORA2BCHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1402900-A1 MEDICINAL COMPOSITIONS Takeda Chemical Industries, Ltd. (JP) 2004-03-31 EP disclosed