SCHEMBL6602974

SCHEMBL6602974

O=C(O)c1cc(OCc2ccccc2)c2cccc(N3CCCCC3)c2n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.44
SLC6A2 P23975 1/20 0.44
SLC6A4 P31645 1/20 0.44
SLC6A3 Q01959 1/20 0.44
NPC1 O15118 1/20 0.44
LMNA P02545 1/20 0.44
POLB P06746 1/20 0.44
MAPT P10636 1/20 0.44
HPGD P15428 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HRH1 P35367 1/20 0.44
HRH3 Q9Y5N1 1/20 0.44
MRGPRX4 Q96LA9 1/20 0.42
BCHE P06276 2/20 0.41
LRRK2 Q5S007 2/20 0.41
PTGER1 P34995 3/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
HTR6 P50406 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6080488 0.91 SMN1; SMN2 (0.42) HTR1ASLC6A2SLC6A4SLC6A3NPC1
SCHEMBL6602328 0.89 ATR (0.50) NPC1MAPTRAB9ALRRK2
SCHEMBL6593434 0.89 ALDH1A1 (0.49) HTR1ASLC6A2SLC6A4SLC6A3MAPT
SCHEMBL6592999 0.89 DRD2 (0.48) LMNAPOLBHPGDSMN1; SMN2HIF1A
SCHEMBL6594774 0.88 SMN1; SMN2 (0.46) HTR1ASLC6A2SLC6A4SLC6A3NPC1
SCHEMBL6080127 0.81 ALDH1A1 (0.49) HTR1AMAPTLRRK2MEN1KMT2A
SCHEMBL6596767 0.79 MRGPRX4 (0.47) NPC1MAPTRAB9ASMN1; SMN2MRGPRX4
SCHEMBL6590520 0.79 MRGPRX4 (0.47) MRGPRX4PTGER1MCL1
SCHEMBL6080492 0.79 HRH3 (0.39) HTR1ASLC6A2SLC6A4SLC6A3NPC1
SCHEMBL6080355 0.79 BACE1 (0.49) LMNAPOLBSMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451159-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2004-09-01 EP claimed
WO-2003010146-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2003-02-06 WO claimed
EP-1451159-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2004-09-01 EP disclosed
WO-2003010146-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2003-02-06 WO disclosed