SCHEMBL6603038

SCHEMBL6603038

COC(=O)COc1ccc2ccccc2n1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYSLTR2 Q9NS75 1/20 0.54
CYSLTR1 Q9Y271 1/20 0.54
ALDH1A1 P00352 5/20 0.50
SMN1; SMN2 Q16637 3/20 0.50
KDM4E B2RXH2 3/20 0.50
HPGD P15428 2/20 0.47
MAPT P10636 4/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
LMNA P02545 1/20 0.45
ALOX15 P16050 1/20 0.45
MAPK1 P28482 1/20 0.45
HSD17B10 Q99714 1/20 0.45
RXFP1 Q9HBX9 1/20 0.45
NOTUM Q6P988 1/20 0.45
POLB P06746 1/20 0.44
GAA P10253 1/20 0.44
ALOX5AP P20292 2/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6601697 0.85 ALDH1A1 (0.70) CYSLTR2CYSLTR1ALDH1A1SMN1; SMN2KDM4E
Benzene SCHEMBL6364361 0.82 MEN1 (0.66) CYSLTR2CYSLTR1ALDH1A1SMN1; SMN2KDM4E
SCHEMBL1495919 0.82 MEN1 (0.66) CYSLTR2CYSLTR1ALDH1A1SMN1; SMN2KDM4E
SCHEMBL8355619 0.81 LTB4R (0.56) CYSLTR2CYSLTR1MAPTMEN1KMT2A
SCHEMBL6608386 0.81 KDM4E (0.52) ALDH1A1SMN1; SMN2KDM4EMAPTMEN1
SCHEMBL6604313 0.80 SMN1; SMN2 (0.48) ALDH1A1SMN1; SMN2KDM4EHPGDMAPT
SCHEMBL29222762 0.78 KDM4E (0.45) CYSLTR2CYSLTR1ALDH1A1SMN1; SMN2KDM4E
Acetone SCHEMBL27714910 0.78 KMT2A (0.49) CYSLTR2CYSLTR1ALDH1A1SMN1; SMN2KDM4E
SCHEMBL6605120 0.77 ALDH1A1 (0.53) CYSLTR2CYSLTR1ALDH1A1SMN1; SMN2KDM4E
SCHEMBL16449538 0.77 KMT2A (0.48) CYSLTR2CYSLTR1ALDH1A1SMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1412349-A2 PIPERAZINE OXYQUINOLINE (NAPHTHALINE) PLATELET ADENOSINE DIPHOSPHATE RECEPTOR ANTAGONISTS Schering Aktiengesellschaft (DE) 2004-04-28 EP claimed
WO-2002098856-A2 PIPERAZINE OXYQUINOLINE (NAPHTHALINE) PLATELET ADENOSINE DIPHOSPHATE RECEPTOR ANTAGONISTS SCHERING AKTIENGESELLSCHAFT (DE) 2002-12-12 WO claimed
US-5488027-A Herbicide-safener combinations containing sulfonylurea or imidazolinone herbicides HOECHST AKTIENGESELLSCHAFT (DE) 1996-01-30 US disclosed