SCHEMBL6603058

SCHEMBL6603058

N=C(NC(=O)c1ccccc1)c1ccc(N2CC(CN3CCN(CCC(=O)OCc4ccccc4)CC3)OC2=O)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 9/20 0.44
ITGA2B P08514 9/20 0.44
SIGMAR1 Q99720 7/20 0.41
PRSS1 P07477 8/20 0.40
PRSS2 P07478 8/20 0.40
PRSS3 P35030 8/20 0.40
F10 P00742 6/20 0.38
GRM2 Q14416 1/20 0.38
SLC6A2 P23975 2/20 0.38
HRH2 P25021 2/20 0.38
HRH1 P35367 2/20 0.38
TMEM97 Q5BJF2 2/20 0.38
CHRM1 P11229 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
HTR1A P08908 1/20 0.37
CHRM5 P08912 1/20 0.37
ADRA1D P25100 1/20 0.37
HTR1B P28222 1/20 0.37
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6601617 0.93 ITGB3 (0.41) ITGB3ITGA2BSIGMAR1PRSS1PRSS2
SCHEMBL6602131 0.93 ITGB3 (0.45) ITGB3ITGA2BSIGMAR1PRSS1PRSS2
SCHEMBL6601020 0.93 ITGB3 (0.41) ITGB3ITGA2BSIGMAR1PRSS1PRSS2
SCHEMBL6604885 0.93 ITGB3 (0.41) ITGB3ITGA2BSIGMAR1SLC6A2HRH2
SCHEMBL6600611 0.92 ITGB3 (0.42) ITGB3ITGA2BSIGMAR1PRSS1PRSS2
SCHEMBL6605994 0.92 ITGB3 (0.48) ITGB3ITGA2BSIGMAR1PRSS1PRSS2
SCHEMBL6601558 0.92 ITGB3 (0.53) ITGB3ITGA2BSIGMAR1PRSS1PRSS2
SCHEMBL6601642 0.92 SIGMAR1 (0.41) ITGB3ITGA2BSIGMAR1PRSS1PRSS2
SCHEMBL6603444 0.91 ITGB3 (0.54) ITGB3ITGA2BSIGMAR1PRSS1PRSS2
SCHEMBL6601675 0.91 ITGB3 (0.54) ITGB3ITGA2BSIGMAR1PRSS1PRSS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0741133-B1 Adhesion receptor antagonists MERCK PATENT GMBH (DE) 2004-01-28 EP disclosed
EP-0741133-A2 Adhesion receptor antagonists MERCK PATENT GmbH (DE) 1996-11-06 EP disclosed