SCHEMBL6604329

SCHEMBL6604329

COc1ccc(SC)c(C2CCN(C(=O)OCc3ccccc3)CC2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.52
NPC1 O15118 2/20 0.52
RAB9A P51151 2/20 0.52
CYP2C19 P33261 1/20 0.50
MMP1 P03956 2/20 0.49
MMP3 P08254 2/20 0.49
MMP7 P09237 2/20 0.49
MMP9 P14780 2/20 0.49
MMP2 P08253 1/20 0.49
MMP8 P22894 1/20 0.49
PDE4B Q07343 1/20 0.48
HTT P42858 1/20 0.48
PRNP P04156 1/20 0.47
GRIN2B Q13224 2/20 0.47
CHRM2 P08172 1/20 0.47
CHRM1 P11229 1/20 0.47
ALDH1A1 P00352 1/20 0.46
SCN5A Q14524 1/20 0.46
SCN9A Q15858 1/20 0.46
TP53 P04637 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6603252 0.92 SMN1; SMN2 (0.52) SMN1; SMN2NPC1RAB9ACYP2C19MMP1
SCHEMBL7669575 0.87 SMN1; SMN2 (0.53) SMN1; SMN2NPC1RAB9ACYP2C19PDE4B
SCHEMBL8316661 0.86 PDE4B (0.58) SMN1; SMN2NPC1RAB9ACYP2C19MMP1
SCHEMBL6613095 0.86 SMN1; SMN2 (0.60) SMN1; SMN2NPC1RAB9ACYP2C19PDE4B
SCHEMBL6710920 0.84 ALDH1A1 (0.56) SMN1; SMN2NPC1RAB9ACYP2C19MMP1
SCHEMBL6605018 0.82 SMN1; SMN2 (0.55) SMN1; SMN2NPC1RAB9ACYP2C19PDE4B
SCHEMBL6608494 0.82 SMN1; SMN2 (0.50) SMN1; SMN2NPC1RAB9ACYP2C19MMP1
SCHEMBL7672654 0.82 PDE4B (0.63) SMN1; SMN2NPC1RAB9ACYP2C19PDE4B
SCHEMBL7669298 0.81 MMP1 (0.54) SMN1; SMN2NPC1RAB9ACYP2C19MMP1
SCHEMBL6603778 0.80 SMN1; SMN2 (0.53) SMN1; SMN2NPC1RAB9ACYP2C19PDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1119551-B1 NAPHTHALENECARBOXAMIDES AS TACHYKININ RECEPTOR ANTAGONISTS ASTRAZENECA AB (SE) 2004-12-29 EP disclosed
EP-1433783-A2 Naphthalenecarboxamides as tachykinin receptor antagonists AstraZeneca AB (SE) 2004-06-30 EP disclosed