SCHEMBL6606975

SCHEMBL6606975

COc1ncc(/C(C#N)=C/c2c(Cl)cncc2Cl)cc1O[C@@H]1CC[C@@H](O)C1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 2/20 0.35
PDE4A P27815 3/20 0.34
PDE4B Q07343 3/20 0.34
PDE4C Q08493 3/20 0.34
PDE4D Q08499 3/20 0.34
ABCB1 P08183 1/20 0.33
ABCG2 Q9UNQ0 1/20 0.33
RECQL P46063 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HIF1A Q16665 1/20 0.33
EGFR P00533 1/20 0.33
PDGFRB P09619 1/20 0.33
PDGFRA P16234 1/20 0.33
IRAK4 Q9NWZ3 1/20 0.31
SCN5A Q14524 2/20 0.31
SCN9A Q15858 2/20 0.31
PRKCQ Q04759 1/20 0.30
PRKCD Q05655 1/20 0.30
KDM4E B2RXH2 1/20 0.30
NPC1 O15118 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6609424 1.00 CHEK1 (0.35) CHEK1PDE4APDE4BPDE4CPDE4D
SCHEMBL6605361 0.89 PDE4D (0.43) CHEK1PDE4APDE4BPDE4CPDE4D
SCHEMBL6605364 0.89 PDE4D (0.43) CHEK1PDE4APDE4BPDE4CPDE4D
SCHEMBL6611995 0.85 PDE4D (0.39) CHEK1PDE4APDE4BPDE4CPDE4D
SCHEMBL6611998 0.85 PDE4D (0.39) CHEK1PDE4APDE4BPDE4CPDE4D
SCHEMBL6607223 0.84 PDE4B (0.38) PDE4APDE4BPDE4CPDE4DRECQL
SCHEMBL6607216 0.84 PDE4B (0.38) PDE4APDE4BPDE4CPDE4DRECQL
SCHEMBL6610689 0.83 CHEK1 (0.36) CHEK1PDE4APDE4BPDE4CPDE4D
SCHEMBL6608573 0.83 PDE4A (0.48) PDE4APDE4BPDE4CPDE4DRECQL
SCHEMBL6609780 0.82 PDE4B (0.44) PDE4APDE4BPDE4CPDE4DABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0882714-B1 SUBSTITUTED VINYLPYRIDINE DERIVATIVES AND DRUGS CONTAINING THE SAME SS PHARMACEUTICAL CO (JP) 2004-03-03 EP disclosed
EP-0882714-A1 SUBSTITUTED VINYLPYRIDINE DERIVATIVES AND DRUGS CONTAINING THE SAME SS Pharmaceutical Co., Ltd. (JP) 1998-12-09 EP disclosed