SCHEMBL6606978

SCHEMBL6606978

COc1ccc(C2=NN(C(=O)c3ccc(NC(=O)c4cnccn4)cc3)CCC2)cc1OC

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CFTR P13569 8/20 0.49
KMT2A Q03164 2/20 0.47
MAOB P27338 1/20 0.46
ALDH1A1 P00352 3/20 0.46
POLB P06746 1/20 0.46
PGR P06401 2/20 0.45
HPGD P15428 1/20 0.45
ABCG2 Q9UNQ0 1/20 0.45
LMNA P02545 2/20 0.45
MEN1 O00255 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.44
KDM4E B2RXH2 1/20 0.44
TP53 P04637 1/20 0.44
MAPT P10636 1/20 0.44
HTT P42858 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
GAA P10253 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6602654 0.94 RAB9A (0.47) CFTRKMT2AALDH1A1POLBPGR
SCHEMBL6600453 0.93 NPC1 (0.47) CFTRKMT2AALDH1A1POLBPGR
SCHEMBL6600681 0.92 PDE4D (0.47) CFTRKMT2AALDH1A1POLBLMNA
SCHEMBL6602109 0.91 RAB9A (0.53) CFTRKMT2AMAOBALDH1A1POLB
SCHEMBL6603519 0.90 MEN1 (0.45) CFTRKMT2AALDH1A1POLBPGR
SCHEMBL6601572 0.90 NPC1 (0.56) CFTRMAOBALDH1A1POLBPGR
SCHEMBL6601859 0.89 CFTR (0.50) CFTRKMT2AMAOBALDH1A1POLB
SCHEMBL147544 0.87 LMNA (0.51) KMT2AMAOBALDH1A1POLBABCG2
SCHEMBL6603307 0.87 LMNA (0.54) CFTRKMT2AMAOBALDH1A1POLB
Hydrochloric Acid SCHEMBL7650133 0.86 LMNA (0.50) CFTRMAOBALDH1A1POLBABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0922036-B1 ARYLALKANOYL PYRIDAZINES MERCK PATENT GMBH (DE) 2004-03-24 EP disclosed