SCHEMBL6606982

SCHEMBL6606982

COc1cccc(/C(Cl)=C\C#N)c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 8/20 0.65
PDE4B Q07343 8/20 0.65
PDE4C Q08493 8/20 0.65
PDE4D Q08499 8/20 0.65
NPC1 O15118 3/20 0.53
RAB9A P51151 3/20 0.53
CES2 O00748 1/20 0.51
CES1 P23141 1/20 0.51
PARP1 P09874 1/20 0.49
PRSS1 P07477 1/20 0.49
PRSS2 P07478 1/20 0.49
PRSS3 P35030 1/20 0.49
ABCG2 Q9UNQ0 1/20 0.45
CHRM2 P08172 1/20 0.44
CHRM1 P11229 1/20 0.44
CHRM3 P20309 1/20 0.44
ALDH1A1 P00352 1/20 0.44
MAPT P10636 1/20 0.44
PKM P14618 1/20 0.44
XBP1 P17861 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6606983 1.00 PDE4A (0.65) PDE4APDE4BPDE4CPDE4DNPC1
SCHEMBL4823570 0.83 PDE4A (0.90) PDE4APDE4BPDE4CPDE4DNPC1
SCHEMBL5194254 0.81 PDE4A (0.60) PDE4APDE4BPDE4CPDE4DCES2
SCHEMBL5194266 0.81 PDE4A (0.60) PDE4APDE4BPDE4CPDE4DCES2
SCHEMBL5194258 0.81 PDE4A (0.60) PDE4APDE4BPDE4CPDE4DCES2
SCHEMBL11117845 0.80 PDE4A (0.65) PDE4APDE4BPDE4CPDE4DNPC1
SCHEMBL11117847 0.80 PDE4A (0.65) PDE4APDE4BPDE4CPDE4DNPC1
SCHEMBL11290195 0.80 PDE4A (0.65) PDE4APDE4BPDE4CPDE4DNPC1
SCHEMBL4825120 0.79 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DNPC1
SCHEMBL4825122 0.79 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1444010-A2 HETEROAROMATIC CARBOXAMIDE DERIVATIVES FOR THE TREATMENT OF INFLAMMATION Pharmacia Corporation (US) 2004-08-11 EP disclosed
WO-2003037886-A2 HETEROAROMATIC CARBOXAMIDE DERIVATIVES FOR THE TREATMENT OF INFLAMMATION PHARMACIA CORPORATION (US) 2003-05-08 WO disclosed