SCHEMBL6607020

SCHEMBL6607020

Cc1nc(-c2ccc(C(F)(F)F)cc2)sc1C(=O)Nc1cccc(OCCN(C(C)C)C(C)C)c1

nearest known ligand 0.62

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 1/20 0.62
PPARA Q07869 10/20 0.53
NPC1 O15118 1/20 0.52
ALDH1A1 P00352 1/20 0.52
GAA P10253 1/20 0.52
MAPT P10636 3/20 0.52
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
MCHR1 Q99705 3/20 0.51
PPARG P37231 3/20 0.47
PPARD Q03181 3/20 0.47
POLB P06746 1/20 0.44
CLK1 P49759 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6603223 0.93 KMT2A (0.58) NR1H4PPARANPC1ALDH1A1GAA
SCHEMBL6604450 0.90 ROCK1 (0.54) NR1H4NPC1MAPTMEN1KMT2A
SCHEMBL6606883 0.90 PARP1 (0.51) NR1H4NPC1ALDH1A1GAAMAPT
SCHEMBL6602401 0.89 MAPT (0.51) NR1H4PPARANPC1GAAMAPT
SCHEMBL6607030 0.89 NR1H4 (0.62) NR1H4PPARANPC1ALDH1A1GAA
SCHEMBL6605510 0.85 MCHR1 (0.67) NR1H4PPARANPC1ALDH1A1GAA
SCHEMBL6603227 0.81 MAPT (0.58) NR1H4PPARANPC1ALDH1A1GAA
SCHEMBL6603148 0.80 MCHR1 (0.65) NR1H4PPARAALDH1A1MAPTMEN1
SCHEMBL6604744 0.78 MCHR1 (0.57) NR1H4PPARANPC1ALDH1A1GAA
SCHEMBL2862288 0.78 NR1H4 (0.59) NR1H4PPARANPC1ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1102535-A4 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORP (US) 2004-09-29 EP disclosed
US-6399656-B1 USING A BENZOPYRAN-3-CARBOXAMIDE COMPOUND SMITHKLINE BEECHAM CORPORATION 2002-06-04 US disclosed
EP-1102535-A2 COMPOUNDS AND METHODS SmithKline Beecham Corporation (US) 2001-05-30 EP disclosed
WO-2000006085-A2 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2000-02-10 WO disclosed