SCHEMBL6607590

SCHEMBL6607590

C=CCc1c(CC(=O)O)ccc(Cl)c1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 2/20 0.41
PTGDR Q13258 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.38
CXCL8 P10145 5/20 0.36
CLIC1 O00299 1/20 0.36
CLCN2 P51788 1/20 0.36
CAMK2A Q9UQM7 4/20 0.35
CYP2C9 P11712 1/20 0.35
AKR1B10 O60218 1/20 0.35
UGT1A9 O60656 1/20 0.35
TRPA1 O75762 1/20 0.35
ABCB11 O95342 1/20 0.35
MT-CO2 P00403 1/20 0.35
TTR P02766 1/20 0.35
ALB P02768 1/20 0.35
UGT1A6 P19224 1/20 0.35
UGT1A1 P22309 1/20 0.35
PTGS1 P23219 1/20 0.35
CXCR1 P25024 1/20 0.35
ADRA1A P35348 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7192003 0.78 AKR1B1 (0.44) AKR1B1PTGDR2CXCL8CLIC1CLCN2
SCHEMBL4900831 0.77 CXCL8 (0.50) AKR1B1CXCL8CLIC1CLCN2CAMK2A
Hydrochloric Acid SCHEMBL11408340 0.75 CXCL8 (0.49) AKR1B1CXCL8CLIC1CLCN2CAMK2A
SCHEMBL9792845 0.74 CYP3A4 (0.32) ALDH1A1
SCHEMBL30423273 0.73 DPP4 (0.40) PTGDRPTGDR2CLCN2ALDH1A1
SCHEMBL55504 0.73 AKR1B1 (0.65) AKR1B1CXCL8CLIC1CLCN2CAMK2A
SCHEMBL29397431 0.73 AKR1B1 (0.65) AKR1B1CXCL8CLIC1CLCN2CAMK2A
SCHEMBL1701239 0.73 AKR1B1 (0.65) AKR1B1CXCL8CLIC1CLCN2CAMK2A
SCHEMBL6391049 0.72 PTGDR (0.60) PTGDRPTGDR2CXCL8CYP2C9KEAP1
SCHEMBL11497864 0.72 TDP1 (0.54) AKR1B1CYP2C9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1032561-B1 SUBSTITUTED OXIMES AS NEUROKININ ANTAGONISTS SCHERING CORP (US) 2004-02-11 EP disclosed
EP-1032561-A1 SUBSTITUTED OXIMES AS NEUROKININ ANTAGONISTS SCHERING CORPORATION (US) 2000-09-06 EP disclosed
US-6063926-A HAVING GREATER BIOACTIVITY SCHERING CORPORATION (US) 2000-05-16 US disclosed
WO-1999026924-A1 SUBSTITUTED OXIMES AS NEUROKININ ANTAGONISTS SCHERING CORPORATION (US) 1999-06-03 WO disclosed