SCHEMBL6607858

SCHEMBL6607858

CCCCOC(=O)NC(=N)NC(=O)c1cnn(-c2ccc3ncccc3c2)c1CCC

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.40
MAPT P10636 5/20 0.40
MAPK1 P28482 4/20 0.38
POLB P06746 1/20 0.38
MAPK14 Q16539 6/20 0.37
GAA P10253 2/20 0.37
LMNA P02545 1/20 0.37
EIF2AK4 Q9P2K8 2/20 0.36
ALOX5 P09917 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6610982 0.88 TAS1R3 (0.39) ALDH1A1EIF2AK4ALOX5
SCHEMBL6319630 0.88 ALDH1A1 (0.41) ALDH1A1MAPTMAPK1POLBMAPK14
SCHEMBL4452237 0.84 ALDH1A1 (0.43) ALDH1A1MAPTMAPK1POLBMAPK14
Trifluoroacetic Acid SCHEMBL6321915 0.79 MAPT (0.45) ALDH1A1MAPTMAPK1POLBMAPK14
SCHEMBL5263394 0.78 ALDH1A1 (0.39) ALDH1A1MAPTMAPK1POLBMAPK14
SCHEMBL6314449 0.78 HPGD (0.46) ALDH1A1MAPTMAPK1MAPK14GAA
SCHEMBL6312734 0.78 NR4A3 (0.49) ALDH1A1MAPTMAPK1POLBMAPK14
SCHEMBL7359681 0.78 MALT1 (0.47) MAPTGAA
SCHEMBL4458512 0.77 MALT1 (0.43) LMNAEIF2AK4
Hydrochloric Acid SCHEMBL6313508 0.76 MALT1 (0.42) LMNAEIF2AK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1056729-B1 N-[(SUBSTITUTED FIVE-MEMBERED DI- OR TRIAZA DIUNSATURATED RING)CARBONYL]GUANIDINE DERIVATIVES FOR THE TREATMENT OF ISCHEMIA PFIZER PROD INC (US) 2004-12-29 EP disclosed
EP-1454902-A1 N- (substituted five-membered di-or triaza diunsaturated ring)carbonyl guanidine derivateives for the treatment of ischemia Pfizer Products Inc. (US) 2004-09-08 EP disclosed