SCHEMBL6608090

SCHEMBL6608090

CC1=C(C#N)C(c2cccc(Br)c2)NC(=O)N1C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
MAPT P10636 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
ALDH1A1 P00352 2/20 0.42
ALOX15 P16050 1/20 0.42
ELANE P08246 3/20 0.40
CYP2C9 P11712 2/20 0.40
TSHR P16473 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
KMT2A Q03164 4/20 0.36
MEN1 O00255 3/20 0.36
LMNA P02545 2/20 0.36
KDM4E B2RXH2 1/20 0.36
HTT P42858 1/20 0.36
TDP1 Q9NUW8 1/20 0.35
POLB P06746 2/20 0.35
CCR1 P32246 1/20 0.35
RECQL P46063 1/20 0.35
HDAC4 P56524 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6609236 0.87 ELANE (0.45) ELANECYP2C9TSHRNPSR1TDP1
SCHEMBL6137166 0.86 KMT2A (0.45) SMN1; SMN2ALDH1A1ELANECYP2C9TSHR
SCHEMBL6608283 0.86 ELANE (0.40) L3MBTL1MAPTALDH1A1ALOX15ELANE
SCHEMBL6137082 0.86 TDP1 (0.50) MAPTALDH1A1ELANECYP2C9KMT2A
SCHEMBL6137365 0.86 ELANE (0.40) MAPTSMN1; SMN2ALDH1A1ELANECYP2C9
SCHEMBL6137118 0.86 HTT (0.43) MAPTSMN1; SMN2ALDH1A1ELANECYP2C9
SCHEMBL6609319 0.84 ALDH1A1 (0.46) MAPK1L3MBTL1MAPTALDH1A1ELANE
SCHEMBL6137233 0.84 ELANE (0.39) MAPK1MAPTSMN1; SMN2ALDH1A1ALOX15
SCHEMBL6137331 0.83 ELANE (0.57) MAPTSMN1; SMN2ALDH1A1ELANECYP2C9
SCHEMBL6137183 0.82 ATM (0.50) L3MBTL1MAPTSMN1; SMN2ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1373223-A4 CYANO-SUBSTITUTED DIHYDROPYRIMIDINE COMPOUNDS AND THEIR USE TO TREAT DISEASES BRISTOL MYERS SQUIBB CO (US) 2004-09-29 EP disclosed
EP-1373223-A1 CYANO-SUBSTITUTED DIHYDROPYRIMIDINE COMPOUNDS AND THEIR USE TO TREAT DISEASES Bristol-Myers Squibb Company (US) 2004-01-02 EP disclosed
WO-2002079169-A1 CYANO-SUBSTITUTED DIHYDROPYRIMIDINE COMPOUNDS AND THEIR USE TO TREAT DISEASES BRISTOL-MYERS SQUIBB COMPANY (US) 2002-10-10 WO disclosed