SCHEMBL6608418

SCHEMBL6608418

COc1ccc(/C(C#N)=C/c2c(Cl)cncc2Cl)nc1O[C@@H]1CC[C@@H](O)C1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.35
PDE4B Q07343 7/20 0.33
PDE4D Q08499 6/20 0.33
PDE4A P27815 5/20 0.33
PDE4C Q08493 5/20 0.33
MAPT P10636 2/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
IRAK4 Q9NWZ3 1/20 0.31
ABCB1 P08183 1/20 0.31
ABCG2 Q9UNQ0 1/20 0.31
RECQL P46063 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
HIF1A Q16665 1/20 0.31
EGFR P00533 1/20 0.31
PDGFRB P09619 1/20 0.31
PDGFRA P16234 1/20 0.31
THRB P10828 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6605174 1.00 CHEK1 (0.35) CHEK1PDE4BPDE4DPDE4APDE4C
SCHEMBL6611085 0.89 PDE4D (0.43) PDE4BPDE4DPDE4APDE4C
SCHEMBL6611092 0.89 PDE4D (0.43) PDE4BPDE4DPDE4APDE4C
SCHEMBL6609891 0.84 PDE4D (0.44) CHEK1PDE4BPDE4DPDE4APDE4C
SCHEMBL6609898 0.84 PDE4D (0.44) CHEK1PDE4BPDE4DPDE4APDE4C
SCHEMBL6606526 0.84 PDE4B (0.42) CHEK1PDE4BPDE4DPDE4APDE4C
SCHEMBL6606520 0.84 PDE4B (0.42) CHEK1PDE4BPDE4DPDE4APDE4C
SCHEMBL6610689 0.84 CHEK1 (0.36) CHEK1PDE4BPDE4DPDE4APDE4C
SCHEMBL6609815 0.82 PDE4A (0.46) PDE4BPDE4DPDE4APDE4CALDH1A1
SCHEMBL6606787 0.80 PDE4D (0.42) PDE4BPDE4DPDE4APDE4CMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0882714-B1 SUBSTITUTED VINYLPYRIDINE DERIVATIVES AND DRUGS CONTAINING THE SAME SS PHARMACEUTICAL CO (JP) 2004-03-03 EP disclosed
EP-0882714-A1 SUBSTITUTED VINYLPYRIDINE DERIVATIVES AND DRUGS CONTAINING THE SAME SS Pharmaceutical Co., Ltd. (JP) 1998-12-09 EP disclosed