SCHEMBL6608558

SCHEMBL6608558

COc1ccc(CNS(=O)(=O)c2ccc(CC(=O)O)cc2)cc1

nearest known ligand 0.78

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.76
ALDH1A1 P00352 5/20 0.72
SMN1; SMN2 Q16637 2/20 0.64
LMNA P02545 2/20 0.64
HTT P42858 1/20 0.64
CYP19A1 P11511 1/20 0.62
USP2 O75604 1/20 0.58
EGFR P00533 3/20 0.58
ERBB2 P04626 2/20 0.58
NAMPT P43490 1/20 0.58
PTGDR2 Q9Y5Y4 2/20 0.57
KDM4E B2RXH2 1/20 0.56
POLB P06746 1/20 0.56
OPRK1 P41145 1/20 0.55
CA12 O43570 1/20 0.55
CA1 P00915 1/20 0.55
CA2 P00918 1/20 0.55
CA9 Q16790 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11113173 0.86 ALDH1A1 (0.79) TSHRALDH1A1SMN1; SMN2LMNAHTT
SCHEMBL20981432 0.86 TSHR (1.00) TSHRALDH1A1SMN1; SMN2LMNAHTT
SCHEMBL1279547 0.86 TSHR (1.00) TSHRALDH1A1SMN1; SMN2LMNAHTT
SCHEMBL5455007 0.86 CYP19A1 (0.66) TSHRALDH1A1CYP19A1NAMPTPTGDR2
SCHEMBL6272107 0.84 ALDH1A1 (0.76) TSHRALDH1A1SMN1; SMN2LMNAHTT
SCHEMBL5458079 0.84 KEAP1 (0.69) TSHRALDH1A1SMN1; SMN2LMNAHTT
SCHEMBL120702 0.84 ALDH1A1 (1.00) TSHRALDH1A1SMN1; SMN2LMNAHTT
SCHEMBL3659182 0.84 ALDH1A1 (0.88) TSHRALDH1A1SMN1; SMN2LMNAHTT
SCHEMBL1278961 0.83 TSHR (0.80) TSHRALDH1A1SMN1; SMN2LMNAHTT
SCHEMBL20981395 0.83 TSHR (0.80) TSHRALDH1A1SMN1; SMN2LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451172-A1 THERAPEUTIC ISOQUINOLINE COMPOUNDS AstraZeneca AB (SE) 2004-09-01 EP disclosed
WO-2003037887-A1 THERAPEUTIC ISOQUINOLINE COMPOUNDS ASTRAZENECA AB (SE) 2003-05-08 WO disclosed