SCHEMBL6610191

SCHEMBL6610191

CC(C)(C)OC(=O)C[C@H](N)C(O)COc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.44
CYP2D6 P10635 2/20 0.43
MTNR1A P48039 3/20 0.40
MTNR1B P49286 3/20 0.40
ADRB2 P07550 1/20 0.40
ADRB1 P08588 1/20 0.40
ADRB3 P13945 1/20 0.40
SCN4A P35499 2/20 0.40
PTPN1 P18031 1/20 0.38
MAOA P21397 1/20 0.38
PTGS1 P23219 1/20 0.38
LTA4H P09960 1/20 0.38
CASR P41180 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27885872 1.00 LMNA (0.44) LMNACYP2D6MTNR1AMTNR1BADRB2
SCHEMBL27869528 0.82 TSHR (0.40) CYP2D6
SCHEMBL27869529 0.82 TSHR (0.40) CYP2D6
SCHEMBL3909668 0.81 LMNA (0.49) LMNACYP2D6MTNR1AMTNR1BADRB2
SCHEMBL6610329 0.80 CYP2D6 (0.50) LMNACYP2D6ADRB2ADRB1ADRB3
SCHEMBL77864 0.80 CTSK (0.37) CYP2D6MTNR1AMTNR1B
SCHEMBL13357117 0.79 LMNA (0.44) LMNACYP2D6MTNR1AMTNR1BADRB2
SCHEMBL79263 0.78 MAPT (0.35) CYP2D6MTNR1AMTNR1B
SCHEMBL487416 0.78 MAPT (0.35) CYP2D6MTNR1AMTNR1B
SCHEMBL473148 0.78 MAPT (0.35) CYP2D6MTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1212309-B1 CASPASE INHIBITOR LG CHEM INVESTMENT LTD (KR) 2004-08-18 EP disclosed
US-6747050-B1 INHIBITING THE ACTIVITY OF CASPASES, PREVENTING INFLAMMATION AND APOPTOSIS LG CHEM INVESTMENT LTD. (KR) 2004-06-08 US disclosed
EP-1212309-A4 CASPASE INHIBITOR LG CHEM INVESTMENT LTD (KR) 2002-11-27 EP disclosed
EP-1212309-A1 CASPASE INHIBITOR LG Chem Investment, Ltd. (KR) 2002-06-12 EP disclosed
WO-2001021600-A1 CASPASE INHIBITOR LG CHEM INVESTMENT LTD. (KR) 2001-03-29 WO disclosed
WO-2001021599-A1 CASPASE INHIBITOR LG CHEMICAL LTD. (KR) 2001-03-29 WO disclosed