SCHEMBL6610643

SCHEMBL6610643

O=C1C(Cc2ccccc2)NC(=O)C2(CCN(CCCCCCc3ccccc3)CC2)N1Cc1ccco1

nearest known ligand 0.59

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 17/20 0.59
CXCR4 P61073 2/20 0.58
CXCR3 P49682 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6610536 0.99 CCR5 (0.57) CCR5CXCR4CXCR3
SCHEMBL6610993 0.96 CXCR3 (0.54) CCR5CXCR4CXCR3
SCHEMBL2086195 0.92 CXCR3 (0.59) CCR5CXCR4CXCR3
SCHEMBL6610890 0.90 CCR5 (0.55) CCR5CXCR4CXCR3
SCHEMBL6611777 0.90 CCR5 (0.55) CCR5CXCR4CXCR3
SCHEMBL6610099 0.90 CCR5 (0.74) CCR5CXCR4
SCHEMBL6613793 0.90 CCR5 (0.52) CCR5CXCR4CXCR3
SCHEMBL6612607 0.89 CCR5 (0.66) CCR5CXCR4CXCR3
SCHEMBL6613597 0.89 CCR5 (0.66) CCR5CXCR4CXCR3
SCHEMBL6616542 0.89 CCR5 (0.73) CCR5CXCR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1236726-B1 TRIAZASPIRO 5.5]UNDECANE DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO (JP) 2004-12-01 EP disclosed
EP-1236726-A1 TRIAZASPIRO 5.5]UNDECANE DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2002-09-04 EP disclosed