SCHEMBL6611673

SCHEMBL6611673

N#Cc1cccc(OCCC2CCCCN2)c1

nearest known ligand 0.72

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 5/20 0.50
CHRNB4 P30926 1/20 0.49
CHRNA3 P32297 1/20 0.49
SLC6A4 P31645 1/20 0.47
HRH1 P35367 1/20 0.44
CCR3 P51677 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11447605 0.96 CHRNB4 (0.53) LTA4HCHRNB4CHRNA3SLC6A4HRH1
SCHEMBL14578215 0.86 CHRNB4 (0.52) LTA4HCHRNB4CHRNA3
SCHEMBL11459383 0.85 LTA4H (0.52) LTA4HSLC6A4
SCHEMBL8290264 0.84 CHRNB4 (0.68) LTA4HCHRNB4CHRNA3
SCHEMBL9237631 0.84 CHRNB4 (0.68) LTA4HCHRNB4CHRNA3
SCHEMBL4965391 0.83 LTA4H (0.64) LTA4H
Hydrochloric Acid SCHEMBL9241805 0.83 CHRNB4 (0.67) LTA4HCHRNB4CHRNA3
Hydrochloric Acid SCHEMBL9241795 0.83 CHRNB4 (0.67) LTA4HCHRNB4CHRNA3
SCHEMBL11447769 0.82 KDM4E (0.49) LTA4HCHRNB4CHRNA3
SCHEMBL11455586 0.82 CHRNB4 (0.69) LTA4HCHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1435955-A2 N-AROYL CYCLIC AMINE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS SmithKline Beecham P.L.C. (GB) 2004-07-14 EP disclosed
WO-2002089800-A2 N-AROYL CYCLIC AMINE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM P.L.C. (GB) 2002-11-14 WO disclosed
US-4225608-A ANTIDEPRESSANTS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1980-09-30 US disclosed