SCHEMBL6614901

SCHEMBL6614901

O=C1C(COCc2ccccc2)NC(=O)C2(CCN(c3ccccc3)CC2)N1Cc1ccco1

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 17/20 0.45
CXCR3 P49682 1/20 0.40
ALDH1A1 P00352 2/20 0.37
USP2 O75604 1/20 0.37
CYP2D6 P10635 1/20 0.37
TSHR P16473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6616504 0.89 CXCR3 (0.51) CCR5CXCR3ALDH1A1USP2CYP2D6
SCHEMBL6612757 0.89 CCR5 (0.56) CCR5CXCR3
SCHEMBL6618118 0.88 CCR5 (0.48) CCR5CXCR3
SCHEMBL6611362 0.87 CCR5 (0.53) CCR5CXCR3ALDH1A1USP2CYP2D6
SCHEMBL6612740 0.86 CCR5 (0.51) CCR5CXCR3
SCHEMBL6612389 0.85 CCR5 (0.54) CCR5CXCR3
SCHEMBL6610890 0.85 CCR5 (0.55) CCR5CXCR3
SCHEMBL6611777 0.85 CCR5 (0.55) CCR5CXCR3
SCHEMBL6611373 0.83 CCR5 (0.61) CCR5CYP2D6
SCHEMBL6611728 0.83 CCR5 (0.47) CCR5CXCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1236726-B1 TRIAZASPIRO 5.5]UNDECANE DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO (JP) 2004-12-01 EP disclosed
EP-1236726-A1 TRIAZASPIRO 5.5]UNDECANE DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2002-09-04 EP disclosed