SCHEMBL6615352

SCHEMBL6615352

CS(=O)(=O)N1Cc2cc(-c3ccncc3)ccc2N(C(=O)C(F)(F)F)CC1Cc1ccccc1

nearest known ligand 0.62

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FNTA P49354 14/20 0.62
FNTB P49356 14/20 0.62
GPR142 Q7Z601 2/20 0.40
DAGLB Q8NCG7 1/20 0.37
DAGLA Q9Y4D2 1/20 0.37
CA1 P00915 2/20 0.37
CA2 P00918 2/20 0.37
CA4 P22748 2/20 0.37
CA9 Q16790 2/20 0.37
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6633140 0.86 FNTA (0.47) FNTAFNTBDAGLBDAGLACYP11B1
SCHEMBL6635731 0.85 FNTA (0.56) FNTAFNTBCA1CA2CA4
SCHEMBL6616410 0.79 CYP11B2 (0.52) FNTAFNTBDAGLBCYP11B1CYP11B2
SCHEMBL3498710 0.76 FNTA (0.73) FNTAFNTB
SCHEMBL3498707 0.76 FNTA (0.73) FNTAFNTB
SCHEMBL6613663 0.76 FNTA (0.62) FNTAFNTBGPR142DAGLBDAGLA
SCHEMBL6637542 0.76 FNTA (0.62) FNTAFNTBGPR142DAGLBDAGLA
SCHEMBL6635023 0.73 FNTA (0.49) FNTAFNTB
SCHEMBL6623755 0.72 FNTA (0.58) FNTAFNTB
SCHEMBL6623752 0.72 FNTA (0.58) FNTAFNTB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1481975-A1 Inhibitors of farnesyl protein transferase BRISTOL-MYERS SQUIBB COMPANY (US) 2004-12-01 EP disclosed
EP-0892797-A4 INHIBITORS OF FARNESYL PROTEIN TRANSFERASE BRISTOL MYERS SQUIBB CO (US) 2004-10-20 EP disclosed
US-6455523-B1 ADMINISTERING 1,4-BENZODIAZEPINE DERIVATIVE AS ANTITUMOR OR ANTICARCINOGENIC AGENT BRISTOL-MYERS SQUIBB COMPANY 2002-09-24 US disclosed
US-6011029-A BENZODIAZEPINE COMPOUNDS BRISTOL-MYERS SQUIBB COMPANY (US) 2000-01-04 US disclosed
EP-0892797-A1 INHIBITORS OF FARNESYL PROTEIN TRANSFERASE BRISTOL-MYERS SQUIBB COMPANY (US) 1999-01-27 EP disclosed
WO-1997030992-A1 INHIBITORS OF FARNESYL PROTEIN TRANSFERASE BRISTOL-MYERS SQUIBB COMPANY (US) 1997-08-28 WO disclosed