SCHEMBL6616613

SCHEMBL6616613

COC(=O)c1cc(CCBr)c2ccccc2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AMPD3 Q01432 1/20 0.48
PPARG P37231 3/20 0.44
PPARA Q07869 3/20 0.44
ALDH1A1 P00352 2/20 0.43
HPGD P15428 2/20 0.43
KDM4E B2RXH2 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
MAPK8 P45983 3/20 0.43
MAPK9 P45984 3/20 0.43
MAPK10 P53779 3/20 0.43
TSHR P16473 1/20 0.42
ATM Q13315 1/20 0.42
LCK P06239 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
CA14 Q9ULX7 1/20 0.41
GPR84 Q9NQS5 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL244415 0.88 HPGD (0.46) AMPD3PPARGPPARAALDH1A1HPGD
SCHEMBL12419947 0.85 HPGD (0.48) AMPD3PPARGPPARAALDH1A1HPGD
SCHEMBL2129601 0.77 ALDH1A1 (0.49) ALDH1A1HPGDKDM4ENPSR1TSHR
SCHEMBL2831563 0.77 HPGD (0.43) AMPD3ALDH1A1HPGDKDM4ENPSR1
SCHEMBL13104720 0.75 ALDH1A1 (0.50) PPARAALDH1A1HPGDKDM4ENPSR1
SCHEMBL161776 0.75 LMNA (0.56) ALDH1A1HPGDKDM4ENPSR1TSHR
SCHEMBL15936293 0.75 ALDH1A1 (0.58) ALDH1A1HPGDKDM4ENPSR1TSHR
SCHEMBL161775 0.75 ALDH1A1 (0.50) ALDH1A1HPGDKDM4ENPSR1TSHR
SCHEMBL19358734 0.75 ALDH1A1 (0.50) ALDH1A1HPGDKDM4ENPSR1TSHR
Bromide SCHEMBL1440188 0.75 ALDH1A1 (0.47) ALDH1A1HPGDKDM4ENPSR1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0683781-B1 NOVEL INHIBITORS OF ADENOSINE MONOPHOSPHATE DEAMINASE METABASIS THERAPEUTICS INC (US) 2004-04-21 EP disclosed
US-5731432-A Inhibitors of adenosine monophosphate deaminase GENSIA SICOR INC. (US) 1998-03-24 US disclosed
EP-0683781-A4 NOVEL INHIBITORS OF ADENOSINE MONOPHOSPHATE DEAMINASE. GENSIA PHARMA (US) 1997-05-28 EP disclosed
EP-0683781-A1 NOVEL INHIBITORS OF ADENOSINE MONOPHOSPHATE DEAMINASE GENSIA PHARMACEUTICALS, INC. (US) 1995-11-29 EP disclosed
WO-1994018200-A1 NOVEL INHIBITORS OF ADENOSINE MONOPHOSPHATE DEAMINASE GENSIA, INC. (US) 1994-08-18 WO disclosed