SCHEMBL6617670

SCHEMBL6617670

O/N=C\c1ccc2c(c1)CCN2C1CCN(CCc2ccc(F)cc2)CC1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.45
HTR2C P28335 3/20 0.45
HTR7 P34969 3/20 0.45
HTR6 P50406 2/20 0.45
NOS3 P29474 1/20 0.39
NOS1 P29475 1/20 0.39
NOS2 P35228 1/20 0.39
HTR1A P08908 1/20 0.38
HTR1D P28221 1/20 0.38
HTR1B P28222 1/20 0.38
HTR1F P30939 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6617673 1.00 HTR2A (0.45) HTR2AHTR2CHTR7HTR6NOS3
SCHEMBL5871718 0.94 HTR1A (0.44) HTR2AHTR2CHTR7HTR6HTR1A
SCHEMBL5871712 0.94 HTR1A (0.44) HTR2AHTR2CHTR7HTR6HTR1A
SCHEMBL5871207 0.84 OPRM1 (0.41) HTR2AHTR2CNOS3NOS1NOS2
SCHEMBL5871211 0.84 OPRM1 (0.41) HTR2AHTR2CNOS3NOS1NOS2
SCHEMBL5871499 0.81 HTR2A (0.40) HTR2AHTR2CHTR7HTR6HTR1A
SCHEMBL5871502 0.81 HTR2A (0.40) HTR2AHTR2CHTR7HTR6HTR1A
SCHEMBL5871325 0.80 HTR1A (0.46) HTR2AHTR2CHTR7HTR6HTR1A
SCHEMBL5870975 0.79 HTR1A (0.55) HTR2AHTR2CHTR1A
SCHEMBL5871190 0.79 SCD (0.52) HTR2AHTR2CHTR7HTR6HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0976732-B1 1,4-SUBSTITUTED CYCLIC AMINE DERIVATIVES EISAI CO LTD (JP) 2004-11-24 EP disclosed