SCHEMBL6618154

SCHEMBL6618154

O=CC1=C(Br)CCc2cc3c(cc21)OCO3

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.45
ALDH1A1 P00352 1/20 0.40
HSD17B10 Q99714 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
ACHE P22303 1/20 0.38
CYP2D6 P10635 2/20 0.38
LMNA P02545 1/20 0.36
HPGD P15428 1/20 0.36
DRD1 P21728 1/20 0.35
DRD5 P21918 1/20 0.35
IDO1 P14902 1/20 0.35
CYP3A4 P08684 1/20 0.34
TSHR P16473 1/20 0.34
CYP2C19 P33261 1/20 0.34
XBP1 P17861 2/20 0.34
METTL3 Q86U44 1/20 0.34
METTL14 Q9HCE5 1/20 0.34
MIF P14174 1/20 0.34
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3267572 0.74
SCHEMBL6336267 0.71 KDM4E (0.58) KDM4EHSD17B10ACHECYP2D6DRD1
SCHEMBL30390377 0.71 KDM4E (0.58) KDM4EHSD17B10ACHECYP2D6DRD1
SCHEMBL16400955 0.70 SRD5A1 (0.49) ALDH1A1TDP1
SCHEMBL3268773 0.68 F7 (0.44) ALDH1A1TDP1
SCHEMBL3272388 0.68 CYP11B2 (0.42)
SCHEMBL21122868 0.68 PARP10 (0.44) ALDH1A1TDP1ACHEMIF
SCHEMBL3267546 0.68 SRD5A1 (0.46) ALDH1A1TDP1
SCHEMBL1243316 0.65 KDM4E (0.54) KDM4EALDH1A1HSD17B10ACHECYP2D6
SCHEMBL1243457 0.65 KDM4E (0.54) KDM4EALDH1A1TDP1ACHECYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1042294-B1 HETEROCYCLIC CYTOTOXIC AGENTS UNIV RUTGERS (US) 2004-08-11 EP disclosed
US-6486167-B1 Heterocyclic cytotoxic agents RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY 2002-11-26 US disclosed
EP-1042294-A1 HETEROCYCLIC CYTOTOXIC AGENTS RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2000-10-11 EP disclosed
WO-1999031067-A1 HETEROCYCLIC CYTOTOXIC AGENTS RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 1999-06-24 WO disclosed