SCHEMBL6618657

SCHEMBL6618657

COc1ccc(-c2ccnn2CC(=O)O)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.50
ALDH1A1 P00352 6/20 0.50
PTGS2 P35354 2/20 0.49
GAA P10253 5/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
PTGS1 P23219 1/20 0.46
PDE3A Q14432 1/20 0.46
HPGD P15428 3/20 0.44
MAPT P10636 2/20 0.44
ALOX15 P16050 2/20 0.44
CASP1 P29466 2/20 0.44
HSD17B10 Q99714 2/20 0.44
LMNA P02545 3/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
USP2 O75604 1/20 0.43
POLB P06746 1/20 0.43
ALOX12 P18054 1/20 0.43
CASP7 P55210 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6651699 0.83 NPC1 (0.48) KDM4EALDH1A1GAAHPGDMAPT
SCHEMBL6497228 0.81 ALDH1A1 (0.55) KDM4EALDH1A1PTGS2HPGDMAPT
SCHEMBL15156844 0.81 HSD17B10 (0.47) KDM4EALDH1A1PTGS2L3MBTL1HPGD
SCHEMBL14973090 0.77 MAPT (0.53) ALDH1A1PTGS2MAPTALOX15HSD17B10
SCHEMBL5285522 0.75 KDM4E (0.53) KDM4EALDH1A1GAAHPGDMAPT
SCHEMBL14351822 0.74 ATM (0.61) KDM4EALDH1A1PTGS2GAAL3MBTL1
SCHEMBL16597364 0.74 PRMT5 (0.52) KDM4EALDH1A1GAAMAPTALOX15
SCHEMBL4483861 0.73 BACE1 (0.61) KDM4EALDH1A1GAAL3MBTL1HPGD
SCHEMBL5647642 0.73 KDM4E (0.51) KDM4EALDH1A1PTGS2GAAL3MBTL1
SCHEMBL5966725 0.72 ALDH1A1 (0.68) ALDH1A1PTGS2HPGDHSD17B10LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1485379-A1 BETA 3-ADRENERGIC RECEPTOR AGONISTS Pfizer Products Inc. (US) 2004-12-15 EP disclosed
WO-2003072572-A1 BETA3-ADRENERGIC RECEPTOR AGONISTS PFIZER PRODUCTS INC. (US) 2003-09-04 WO disclosed