SCHEMBL6621186

SCHEMBL6621186

COc1ccc2c(c1)ncc1c3cc(OC)c(OC)cc3ccc21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 4/20 0.51
RAD52 P43351 1/20 0.50
PDGFRB P09619 5/20 0.48
PDGFRA P16234 5/20 0.48
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
EGFR P00533 2/20 0.45
HPGDS O60760 1/20 0.44
PDPK1 O15530 2/20 0.44
GABRA1 P14867 1/20 0.44
GABRG2 P18507 1/20 0.44
GABRB3 P28472 1/20 0.44
GABRA5 P31644 1/20 0.44
GABRA3 P34903 1/20 0.44
GABRA6 Q16445 1/20 0.44
IDO1 P14902 1/20 0.44
TDO2 P48775 1/20 0.44
PDE3B Q13370 1/20 0.44
PDE3A Q14432 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28281503 0.89 PDE10A (0.54) PDE10ARAD52PDGFRBPDGFRAKDM4E
SCHEMBL6631633 0.88 RAD52 (0.53) PDE10ARAD52PDGFRBPDGFRAEGFR
SCHEMBL6616005 0.88 PDPK1 (0.51) PDGFRBPDGFRAALDH1A1SMN1; SMN2PDPK1
SCHEMBL28118851 0.79 RAD52 (0.67) PDE10ARAD52KDM4EALDH1A1SMN1; SMN2
SCHEMBL6615366 0.78 RAB9A (0.51) PDGFRBPDGFRAKDM4EALDH1A1SMN1; SMN2
SCHEMBL6618226 0.77 PDPK1 (0.54) PDE10AKDM4ESMN1; SMN2PDPK1
SCHEMBL30159718 0.77 CA12 (0.56) PDE10ARAD52KDM4EALDH1A1SMN1; SMN2
SCHEMBL28118318 0.77 CA12 (0.56) PDE10ARAD52KDM4EALDH1A1SMN1; SMN2
SCHEMBL1132076 0.77 TDP1 (0.50) KDM4EALDH1A1SMN1; SMN2IDO1TDO2
SCHEMBL6360527 0.77 RAD52 (0.47) PDE10ARAD52PDGFRBPDGFRAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1042294-B1 HETEROCYCLIC CYTOTOXIC AGENTS UNIV RUTGERS (US) 2004-08-11 EP disclosed
US-6486167-B1 Heterocyclic cytotoxic agents RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY 2002-11-26 US disclosed
EP-1042294-A1 HETEROCYCLIC CYTOTOXIC AGENTS RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2000-10-11 EP disclosed
WO-1999031067-A1 HETEROCYCLIC CYTOTOXIC AGENTS RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 1999-06-24 WO disclosed