SCHEMBL6616005

SCHEMBL6616005

COc1cc2ccc3c4cc(OC)c(OC)cc4ncc3c2cc1OC

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 8/20 0.51
DAPK3 O43293 1/20 0.48
PRKD3 O94806 1/20 0.48
FLT1 P17948 1/20 0.48
RPS6KA3 P51812 1/20 0.48
LRRK2 Q5S007 1/20 0.48
PDGFRB P09619 10/20 0.46
PDGFRA P16234 10/20 0.46
ALDH1A1 P00352 1/20 0.46
GLA P06280 1/20 0.46
GAA P10253 1/20 0.46
MAPT P10636 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6631633 0.88 RAD52 (0.53) PDPK1DAPK3PRKD3FLT1RPS6KA3
SCHEMBL6621186 0.88 PDE10A (0.51) PDPK1PDGFRBPDGFRAALDH1A1SMN1; SMN2
SCHEMBL6616039 0.86 TDP1 (0.51) PDPK1ALDH1A1MAPTSMN1; SMN2
SCHEMBL6618226 0.85 PDPK1 (0.54) PDPK1DAPK3PRKD3FLT1RPS6KA3
SCHEMBL1132076 0.85 TDP1 (0.50) ALDH1A1MAPTSMN1; SMN2
SCHEMBL27751211 0.78 ALDH1A1 (0.50) ALDH1A1GAAMAPTSMN1; SMN2
SCHEMBL6617564 0.77 PDGFRB (0.58) PDPK1PDGFRBPDGFRA
SCHEMBL8317211 0.76 NQO2 (0.48) PDGFRBPDGFRAALDH1A1GLAGAA
SCHEMBL28281503 0.75 PDE10A (0.54) PDPK1PDGFRBPDGFRAALDH1A1MAPT
SCHEMBL4745584 0.74 ENPP1 (0.49) PDPK1PDGFRBPDGFRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1042294-B1 HETEROCYCLIC CYTOTOXIC AGENTS UNIV RUTGERS (US) 2004-08-11 EP disclosed
US-6486167-B1 Heterocyclic cytotoxic agents RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY 2002-11-26 US disclosed
US-6140328-A FOR TREATING TUMOR RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2000-10-31 US disclosed
EP-1042294-A1 HETEROCYCLIC CYTOTOXIC AGENTS RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2000-10-11 EP disclosed
WO-1999031067-A1 HETEROCYCLIC CYTOTOXIC AGENTS RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 1999-06-24 WO disclosed