Apronal

Apronal

SCHEMBL662209

C=CCC(C(=O)NC(N)=O)C(C)C

nearest known ligand 0.37

Full drug profile on Sugi Atlas →

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 2/20 0.37
MMP3 P08254 2/20 0.37
MMP7 P09237 2/20 0.37
MMP1 P03956 1/20 0.37
MAPT P10636 1/20 0.36
CACNA1B Q00975 1/20 0.36
APBA1 Q02410 1/20 0.36
ECE1 P42892 3/20 0.33
CRBN Q96SW2 1/20 0.32
GRIK1 P39086 2/20 0.31
GRIK2 Q13002 2/20 0.31
RECQL P46063 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10394988 0.86 TAS2R38 (0.36) MMP2MMP3MMP7MMP1ECE1
Urea SCHEMBL29215668 0.79 SLC1A3 (0.45) MMP2MMP3MMP7MMP1ECE1
SCHEMBL13500189 0.79 MMP2 (0.49) MMP2MMP3MMP7MMP1
SCHEMBL3322985 0.78 GRIK1 (0.35) MMP2MMP3MMP7MMP1ECE1
SCHEMBL13499675 0.77 MMP2 (0.44) MMP2MMP3MMP7MMP1ECE1
SCHEMBL29215667 0.76 MAPT (0.35) MMP2MMP3MMP7MMP1MAPT
SCHEMBL13461535 0.76 MMP2 (0.38) MMP2MMP3MMP7MMP1ECE1
SCHEMBL13435005 0.74 MMP2 (0.43) MMP2MMP3MMP7MMP1ECE1
SCHEMBL3651551 0.73 CA1 (0.45) MAPTECE1CRBN
SCHEMBL3651490 0.73 CA1 (0.45) MAPTECE1CRBN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 466 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118872662-A Ultralow temperature preservation method of umbilical cord blood mononuclear cells and freezing storage liquid set 深圳市中佳生物医疗科技有限公司 2024-11-01 CN claimed
CN-110511141-A A kind of synthetic method of apronal SHANGHAI LINKCHEM TECH CO LTD 2019-11-29 CN claimed
CN-107501129-A A kind of synthetic method of apronal 陕西师范大学 2017-12-22 CN claimed
EP-2702989-B1 STABLE PHARMACEUTICAL COMPOSITION KOWA CO (JP) 2017-08-23 EP claimed
EP-2702989-A1 STABLE PHARMACEUTICAL COMPOSITION Kowa Company, Ltd. (JP) 2014-03-05 EP claimed
US-20120095104-A1 USE OF VASOCONSTRICTORS ZACHAR ORON (IL) 2012-04-19 US claimed
CN-102300566-A Cutaneous application of vasoconstrictors 2011-12-28 CN claimed
EP-2376073-A2 DERMAL APPLICATION OF VASOCONSTRICTORS Zachar, Oron (IL) 2011-10-19 EP claimed
US-20110144209-A1 USE OF VASOCONSTRICTORS ZACHAR ORON 2011-06-16 US claimed
EP-2313037-A1 DERMAL APPLICATION OF VASOCONSTRICTORS Zachar, Oron (IL) 2011-04-27 EP claimed
EP-1073470-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2001-02-07 EP claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed
EP-1027339-A1 METHOD AND REAGENTS FOR N-ALKYLATING UREIDES TARO PHARMACEUTICAL INDUSTRIES LIMITED (IL) 2000-08-16 EP claimed
US-6093820-A REACTING AN IMIDE WITH A (SUBSTITUTED)ALKOXYALKYLSULFONIC ACID ESTER TO FORM A N-ALKOXYALKYL IMIDE SUCH AS METHOXYMETHYL ETHOSUXIMIDE; ADMINISTERING AS ANTICONVULSANT, ANTIANXIETY AGENT AND MUSCLE RELAXANT TARO PHARMACEUTICAL INDUSTRIES LTD. (IL) 2000-07-25 US claimed
WO-1999018084-A1 METHOD AND REAGENTS FOR N-ALKYLATING UREIDES TARO PHARMACEUTICAL INDUSTRIES LTD. (IL) 1999-04-15 WO claimed
US-5686109-A MIXTURE OF IBUPROFEN AND ISOPROPYLANTIPYRINE, REDUCED SIDE EFFECTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-11-11 US claimed
US-5585243-A SEPARATELY INCUBATING HUMAN PLATELETS WITH BLOOD SAMPLE ANDREAGENT DRUG SOLUTION TO FORM COMPLEXES, DETERMINING AMOUNT OF BOUND ANTIBODY THE BLOOD CENTER OF SOUTHEASTERN WISCONSIN, INC. (US) 1996-12-17 US claimed
US-5409709-A Coating a layer of ibuprofen, a layer of magnesium-based antacid and a layer between the above layers of acetaminophen; sustained release; antiinflammatory agent LION CORPORATION (JP) 1995-04-25 US claimed
WO-1995008116-A1 METHOD OF DETECTING CYTOPENIA THAT IS MEDIATED BY DRUG-DEPENDENT ANTIBODY BINDING TO BLOOD CELLS THE BLOOD CENTER OF SOUTHEASTERN WISCONSIN, INC. (US) 1995-03-23 WO claimed
US-4557934-A ALONG WITH A DIOL PYRROLIDONE OR AN AZACYCLOPENTAN-2-ONE THE PROCTER & GAMBLE COMPANY (US) 1985-12-10 US claimed