SCHEMBL6626258

SCHEMBL6626258

COc1cc2c(cc1OC)C(c1ccc(-c3cccc(C(F)(F)F)c3)cc1)=NN(C)C(=O)C2.COc1ccc(-c2ccc(C3=NN(C)C(=O)Cc4cc(OC)c(OC)cc43)cc2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 1/20 0.43
ALDH1A1 P00352 2/20 0.42
LMNA P02545 1/20 0.42
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
MAPK1 P28482 1/20 0.40
CYP2C19 P33261 1/20 0.40
MAOA P21397 2/20 0.40
PDGFRB P09619 1/20 0.39
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39
GRM5 P41594 1/20 0.39
GRM1 Q13255 1/20 0.39
PLAU P00749 2/20 0.39
PLAT P00750 2/20 0.39
PLG P00747 1/20 0.39
NPSR1 Q6W5P4 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
GRIN2C Q14957 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5484469 0.96 CYP1A2 (0.43) NR1H4ALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL5486696 0.87 CYP1A2 (0.47) ALDH1A1LMNACYP1A2CYP3A4CYP2C9
SCHEMBL5492316 0.87 ALDH1A1 (0.53) ALDH1A1LMNACYP1A2CYP3A4CYP2C9
SCHEMBL5486160 0.86 MAPK1 (0.46) ALDH1A1LMNACYP1A2CYP3A4CYP2C9
SCHEMBL5490322 0.82 CYP1A2 (0.46) ALDH1A1LMNACYP1A2CYP3A4CYP2C9
SCHEMBL5492933 0.79 TDP2 (0.47) ALDH1A1CYP1A2CYP3A4CYP2C9MAPK1
SCHEMBL5484921 0.79 CYP1A2 (0.50) ALDH1A1LMNACYP1A2CYP3A4CYP2C9
SCHEMBL5488285 0.78 TDP2 (0.46) LMNACYP1A2CYP3A4CYP2C9MAPK1
SCHEMBL5493764 0.78 MAPK1 (0.49) ALDH1A1LMNACYP1A2CYP3A4CYP2C9
SCHEMBL5484416 0.77 CYP11B1 (0.47) CYP1A2CYP3A4CYP2C9MAPK1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1392663-A2 CYCLIC NUCLEOTIDE PHOSPHODIESTERASE INHIBITORS, PREPARATION AND USES THEREOF NEURO3D (FR) 2004-03-03 EP claimed
WO-2002098865-A2 CYCLIC NUCLEOTIDE PHOSPHODIESTERASE INHIBITORS, PREPARATION AND USES THEREOF NEURO3D (FR) 2002-12-12 WO claimed