SCHEMBL6627378

SCHEMBL6627378

CC(C)(C)OC(=O)NCc1ccnc(OC(=O)O)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.46
BRD4 O60885 1/20 0.44
NAMPT P43490 2/20 0.43
GLS O94925 3/20 0.41
KDM4A O75164 1/20 0.41
HDAC1 Q13547 1/20 0.40
GRM2 Q14416 1/20 0.40
CYP3A4 P08684 1/20 0.40
ACACB O00763 1/20 0.40
ACACA Q13085 1/20 0.40
MAPT P10636 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
RECQL P46063 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
NR1H4 Q96RI1 1/20 0.38
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10165065 0.87 LOX (0.48) L3MBTL1BRD4NAMPTGLSKDM4A
SCHEMBL8226463 0.82 L3MBTL1 (0.44) L3MBTL1BRD4NAMPTGLSKDM4A
SCHEMBL1698559 0.82 L3MBTL1 (0.47) L3MBTL1BRD4NAMPTGLSKDM4A
SCHEMBL29693623 0.82 L3MBTL1 (0.47) L3MBTL1BRD4NAMPTGLSKDM4A
SCHEMBL30400296 0.81 L3MBTL1 (0.43) L3MBTL1BRD4NAMPTGLSKDM4A
SCHEMBL15871964 0.81 BRD4 (0.49) L3MBTL1BRD4NAMPTGLSKDM4A
SCHEMBL30399922 0.81 L3MBTL1 (0.49) L3MBTL1BRD4NAMPTGLSKDM4A
SCHEMBL10163771 0.81 L3MBTL1 (0.49) L3MBTL1BRD4NAMPTGLSKDM4A
SCHEMBL18049277 0.81 LOXL2 (0.60) L3MBTL1BRD4NAMPTHDAC1CYP3A4
SCHEMBL30931637 0.81 EPHX2 (0.44) L3MBTL1BRD4NAMPTGLSKDM4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1392680-A2 SELECTIVE ANTHRANILAMIDE PYRIDINE AMIDES AS INHIBITORS OF VEGFR-2 AND VEGFR-3 SCHERING AKTIENGESELLSCHAFT (DE) 2004-03-03 EP disclosed
WO-2002090352-A2 SELECTIVE ANTHRANILAMIDE PYRIDINE AMIDES AS INHIBITORS OF VEGFR-2 AND VEGFR-3 SCHERING AKTIENGESELLSCHAFT (DE) 2002-11-14 WO disclosed