SCHEMBL6628532

SCHEMBL6628532

CC(C)C[CH]C(=O)N[C@H]1CCCN(S(=O)(=O)c2ccc[n+]([O-])c2)CC1=O

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTSK P43235 13/20 0.43
CTSL P07711 5/20 0.40
CTSS P25774 5/20 0.40
CTSB P07858 3/20 0.39
CTSV O60911 1/20 0.39
TDP1 Q9NUW8 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
ALDH1A1 P00352 1/20 0.34
GAA P10253 1/20 0.34
LMNA P02545 1/20 0.34
MMP3 P08254 1/20 0.34
ADAM17 P78536 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5105882 0.91 CTSK (0.41) CTSKCTSLCTSSCTSBCTSV
SCHEMBL5096573 0.87 EPHX2 (0.42) CTSKCTSLCTSSCTSBCTSV
SCHEMBL5092584 0.87 CTSK (0.47) CTSKCTSLCTSSCTSBCTSV
SCHEMBL4766701 0.86 MEN1 (0.43) CTSKCTSLCTSSCTSBMEN1
SCHEMBL7427478 0.86 MEN1 (0.43) CTSKCTSLCTSSCTSBMEN1
SCHEMBL5093139 0.86 KMT2A (0.45) CTSKTDP1MEN1KMT2AALDH1A1
SCHEMBL7434825 0.86 KMT2A (0.45) CTSKTDP1MEN1KMT2AALDH1A1
SCHEMBL4686403 0.86 CTSK (0.54) CTSKCTSLCTSSCTSBCTSV
SCHEMBL7431349 0.85 KMT2A (0.45) CTSKCTSLCTSSCTSBCTSV
SCHEMBL5096578 0.85 POLB (0.48) CTSKCTSLCTSSCTSBCTSV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1384713-A1 4-amino-azepan-3-one derivatives as protease inhibitors SmithKline Beecham Corporation (US) 2004-01-28 EP disclosed