SCHEMBL7434825

SCHEMBL7434825

CC(C)C[CH]C(=O)NC1CCCN(S(=O)(=O)c2ccc(F)cc2)CC1=O

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.45
MAPT P10636 2/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C19 P33261 1/20 0.44
ALDH1A1 P00352 1/20 0.43
TP53 P04637 1/20 0.43
TDP1 Q9NUW8 1/20 0.42
EPHX2 P34913 1/20 0.41
PKM P14618 1/20 0.41
KDM4E B2RXH2 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CTSK P43235 2/20 0.41
GAA P10253 1/20 0.41
MEN1 O00255 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5093139 1.00 KMT2A (0.45) KMT2AMAPTCYP3A4CYP2C19ALDH1A1
SCHEMBL5096573 0.91 EPHX2 (0.42) KMT2AALDH1A1EPHX2CTSKMEN1
SCHEMBL5092584 0.91 CTSK (0.47) KMT2AALDH1A1TDP1EPHX2CTSK
SCHEMBL5099202 0.91 KMT2A (0.43) KMT2AMAPTCYP3A4CYP2C19ALDH1A1
SCHEMBL4766701 0.90 MEN1 (0.43) KMT2ACTSKGAAMEN1
SCHEMBL7427478 0.90 MEN1 (0.43) KMT2ACTSKGAAMEN1
SCHEMBL5096578 0.89 POLB (0.48) KMT2AMAPTALDH1A1PKMCTSK
SCHEMBL6628532 0.86 CTSK (0.43) KMT2AALDH1A1TDP1CTSKGAA
SCHEMBL7432025 0.86 ALDH1A1 (0.45) KMT2AALDH1A1EPHX2L3MBTL1CTSK
SCHEMBL7434831 0.83 KMT2A (0.48) KMT2AMAPTCYP3A4CYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1158986-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2002-03-27 EP claimed
EP-1158986-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2001-12-05 EP claimed
WO-2000038687-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2000-07-06 WO claimed