SCHEMBL6628971

SCHEMBL6628971

CCCc1ccncc1-c1nc(-c2ccc(C(F)(F)F)cc2)cs1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.51
L3MBTL1 Q9Y468 2/20 0.51
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
ATP4A P20648 3/20 0.48
ATP4B P51164 3/20 0.48
RAB9A P51151 3/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
AR P10275 1/20 0.46
NPC1 O15118 1/20 0.46
SREBF2 Q12772 6/20 0.45
LTA4H P09960 1/20 0.44
CYP19A1 P11511 2/20 0.44
LMNA P02545 2/20 0.43
CDK5 Q00535 1/20 0.43
CDK5R1 Q15078 1/20 0.43
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
ATM Q13315 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6626251 0.92 KDM4E (0.52) KDM4EL3MBTL1MEN1KMT2ANPSR1
SCHEMBL6648508 0.90 KDM4E (0.51) KDM4EL3MBTL1KMT2ARAB9ASMN1; SMN2
SCHEMBL6647939 0.89 SREBF2 (0.41) KDM4EL3MBTL1MEN1KMT2ANPSR1
SCHEMBL6649838 0.86 KDM4E (0.59) KDM4EL3MBTL1RAB9ASMN1; SMN2AR
SCHEMBL6649722 0.85 SREBF2 (0.46) KDM4EMEN1KMT2AATP4AATP4B
SCHEMBL6649085 0.84 KDM4E (0.59) KDM4EL3MBTL1MEN1KMT2ARAB9A
SCHEMBL6649374 0.84 SREBF2 (0.59) KDM4EL3MBTL1MEN1KMT2ARAB9A
SCHEMBL6647164 0.84 KDM4E (0.59) KDM4EL3MBTL1MEN1KMT2ANPSR1
SCHEMBL6649370 0.84 CYP19A1 (0.46) KDM4EL3MBTL1MEN1KMT2ARAB9A
SCHEMBL6650443 0.84 SREBF2 (0.55) KDM4EMEN1KMT2AATP4AATP4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1432706-A2 3-PYRIDYL OR 4-ISOQUINOLINYL THIAZOLES AS C17,20 LYASE INHIBITORS Bayer Pharmaceuticals Corporation (US) 2004-06-30 EP disclosed
WO-2003027085-A2 3-PYRIDYL OR 4-ISOQUINOLINYL THIAZOLES AS C17,20 LYASE INHIBITORS BAYER PHARMACEUTICALS CORPORATION (US) 2003-04-03 WO disclosed