SCHEMBL6629187

SCHEMBL6629187

CCCCCc1ccc2c(c1)-c1c3c(c4c([nH]c5ccccc54)c1C2)C(=O)NC3=O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKD3 O94806 5/20 0.53
PRKCG P05129 5/20 0.53
PRKCB P05771 5/20 0.53
PRKCA P17252 5/20 0.53
PRKCH P24723 5/20 0.53
PRKCI P41743 5/20 0.53
PRKCE Q02156 5/20 0.53
PRKCQ Q04759 5/20 0.53
PRKCZ Q05513 5/20 0.53
PRKCD Q05655 5/20 0.53
PRKD1 Q15139 5/20 0.53
MAP3K9 P80192 3/20 0.53
MAP3K10 Q02779 3/20 0.53
MAP3K11 Q16584 3/20 0.53
DAPK3 O43293 1/20 0.53
PARP1 P09874 5/20 0.49
CHEK1 O14757 3/20 0.48
CDK4 P11802 6/20 0.48
CCND1 P24385 6/20 0.48
NTRK1 P04629 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6630190 0.81 CDK4 (0.62) PRKD3PRKCGPRKCBPRKCAPRKCH
SCHEMBL6630441 0.80 CDK4 (0.63) PRKD3PRKCGPRKCBPRKCAPRKCH
SCHEMBL6632580 0.80 CDK4 (0.63) PRKD3PRKCGPRKCBPRKCAPRKCH
SCHEMBL3075228 0.79 MAP3K9 (0.80) PRKD3PRKCGPRKCBPRKCAPRKCH
SCHEMBL6627743 0.77 PRKD3 (0.65) PRKD3PRKCGPRKCBPRKCAPRKCH
SCHEMBL6629947 0.72 MAP3K9 (0.64) PRKD3PRKCGPRKCBPRKCAPRKCH
SCHEMBL7354146 0.70 MAP3K9 (0.68) PRKD3PRKCGPRKCBPRKCAPRKCH
SCHEMBL6631769 0.70 CDK4 (0.63) PRKD3PRKCGPRKCBPRKCAPRKCH
SCHEMBL6629885 0.70 CDK4 (0.63) PRKD3PRKCGPRKCBPRKCAPRKCH
Staurosporine Aglycon SCHEMBL29406635 0.67 CDK4 (1.00) PRKD3PRKCGPRKCBPRKCAPRKCH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1088823-B1 Fused pyrrolocarbazoles CEPHALON INC (US) 2004-12-29 EP disclosed
EP-0785938-B1 FUSED PYRROLOCARBAZOLES CEPHALON INC (US) 2002-01-02 EP disclosed
US-5594009-A KINASE INHIBITORS, TROPHIC FACTOR-INDUCED ACTIVITY ENHANCEMENT, CELL SURVIVAL CEPHALON, INC. (US) 1997-01-14 US disclosed
US-5591855-A KINASE INHIBITORS, TROPHIC FACTOR-INDUCED ACTIVITY ENHANCEMENT, CELL SURVIVAL CEPHALON, INC. (US) 1997-01-07 US disclosed