SCHEMBL6629207

SCHEMBL6629207

N#CC1(NC(=O)C(COC(=O)N2CCOCC2)S(=O)(=O)Cc2ccccc2)CCOCC1

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSS P25774 16/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
CTSL P07711 9/20 0.43
CTSK P43235 8/20 0.43
CTSB P07858 7/20 0.43
GAA P10253 1/20 0.38
TSHR P16473 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7656008 0.82 CTSS (0.47) CTSSCTSLCTSKCTSB
SCHEMBL6063338 0.81 CTSS (0.44) CTSSMEN1KMT2ANPSR1CTSL
SCHEMBL6063336 0.81 CTSS (0.44) CTSSMEN1KMT2ANPSR1CTSL
SCHEMBL6628713 0.78 CTSS (0.47) CTSSMEN1KMT2ANPSR1CTSL
SCHEMBL6628710 0.78 CTSS (0.47) CTSSMEN1KMT2ANPSR1CTSL
SCHEMBL5955838 0.73 CTSS (0.60) CTSSCTSLCTSKCTSB
SCHEMBL7656003 0.73 CTSS (0.55) CTSSCTSLCTSKCTSB
SCHEMBL7655999 0.73 CTSS (0.55) CTSSCTSLCTSKCTSB
SCHEMBL3907834 0.72 CTSS (0.50) CTSSMEN1KMT2ANPSR1CTSL
SCHEMBL3893947 0.70 CTSS (0.48) CTSSCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1397340-A2 CHEMICAL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS AS CATHEPSIN S INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2004-03-17 EP disclosed
WO-2002098850-A2 CHEMICAL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS AS CATHEPSIN S INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2002-12-12 WO disclosed