SCHEMBL6629360

SCHEMBL6629360

Cc1cc(C)cc(NC(=O)C(Br)C(=O)c2ccccc2)c1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.51
HTT P42858 3/20 0.47
NPSR1 Q6W5P4 2/20 0.47
ATM Q13315 3/20 0.46
RAB9A P51151 3/20 0.46
GAA P10253 3/20 0.46
NPC1 O15118 2/20 0.46
HSP90AA1 P07900 2/20 0.46
TDP1 Q9NUW8 2/20 0.46
ALDH1A1 P00352 4/20 0.44
KMT2A Q03164 4/20 0.42
MEN1 O00255 3/20 0.42
GPR55 Q9Y2T6 1/20 0.42
MAPT P10636 2/20 0.42
LMNA P02545 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
HPGD P15428 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL628191 0.84 GAA (0.64) HTTNPSR1ATMRAB9AGAA
SCHEMBL10875758 0.75 RAB9A (0.65) HTTNPSR1RAB9AGAANPC1
SCHEMBL3274053 0.75 THRB (0.79) THRBHTTRAB9AGAANPC1
SCHEMBL6719393 0.72 TDP1 (0.55) THRBHTTNPSR1GAATDP1
SCHEMBL330776 0.72 TDP1 (0.56) ATMRAB9AGAANPC1HSP90AA1
SCHEMBL11179333 0.72 NPSR1 (0.58) THRBHTTNPSR1GAATDP1
SCHEMBL22173521 0.72 THRB (0.73) THRBHTTRAB9AGAANPC1
SCHEMBL27745059 0.71 KMT2A (0.44) HTTNPSR1ATMRAB9AGAA
Benzamide SCHEMBL28002190 0.71 THRB (0.57) THRBRAB9ANPC1TDP1KMT2A
SCHEMBL6719138 0.71 KMT2A (0.59) THRBHTTNPSR1GAATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1349860-B1 SYNTHESES FOR PREPARING 1,4-DIKETOPYRROLO[3,4-C]PYRROLES SUN CHEMICAL CORP (US) 2004-08-18 EP disclosed
EP-1349860-A2 SYNTHESES FOR PREPARING 1,4-DIKETOPYRROLO[3,4-C]PYRROLES SUN CHEMICAL CORPORATION (US) 2003-10-08 EP disclosed
WO-2002068422-A2 SYNTHESES FOR PREPARING 1,4-DIKETOPYRROLO[3,4-C]PYRROLES SUN CHEMICAL CORPORATION (US) 2002-09-06 WO disclosed
US-6388093-B1 REACTING A B-KETOAMIDE WITH A STRONG BASE; HALOGENTAION; CYCLIZATION SUN CHEMICAL CORPORATION 2002-05-14 US disclosed