SCHEMBL6629375

SCHEMBL6629375

CCc1ncc(-c2ccc(CS)cc2)o1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.45
RXRA P19793 2/20 0.40
RXRB P28702 2/20 0.40
RXRG P48443 2/20 0.40
FFAR1 O14842 1/20 0.36
TSHR P16473 2/20 0.36
ALOX15 P16050 1/20 0.36
CASP1 P29466 1/20 0.36
IDO1 P14902 1/20 0.35
HDAC1 Q13547 4/20 0.35
HDAC2 Q92769 4/20 0.35
HDAC3 O15379 3/20 0.35
HDAC4 P56524 3/20 0.35
HDAC7 Q8WUI4 3/20 0.35
HDAC10 Q969S8 3/20 0.35
HDAC11 Q96DB2 3/20 0.35
HDAC8 Q9BY41 3/20 0.35
HDAC6 Q9UBN7 3/20 0.35
HDAC9 Q9UKV0 3/20 0.35
HDAC5 Q9UQL6 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1617734 0.79 RAB9A (0.51) NOTUMRXRARXRBRXRGTSHR
SCHEMBL7903330 0.79 NOTUM (0.70) NOTUMRXRARXRBRXRGTSHR
SCHEMBL12188072 0.79 NOTUM (0.47) NOTUMRXRARXRBRXRGTSHR
SCHEMBL1696557 0.79 NOTUM (0.68) NOTUMRXRARXRBRXRGFFAR1
SCHEMBL27343825 0.77 NOTUM (0.45) NOTUMRXRARXRBRXRGTSHR
SCHEMBL22556732 0.77 NOTUM (0.49) NOTUMRXRARXRBRXRGFFAR1
SCHEMBL6629373 0.75 NOTUM (0.44) NOTUMRXRARXRBRXRGTSHR
SCHEMBL1617655 0.71 RXRA (0.42) NOTUMRXRARXRBRXRGFFAR1
SCHEMBL5585973 0.71 NOTUM (0.43) NOTUMRXRARXRBRXRGFFAR1
SCHEMBL20747003 0.70 CA12 (0.54) NOTUMTSHRALOX15CASP1HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1394162-A1 Intermediates of azole antifungal agents and processes for the preparation thereof Eisai Co., Ltd. (JP) 2004-03-03 EP disclosed
EP-1394142-A1 Carboxylic acid intermediates of antifungal agents and processes for the preparation thereof Eisai Co., Ltd. (JP) 2004-03-03 EP disclosed
EP-1231210-A2 Azole antifungal agents, processes for the preparation thereof, and intermediates Eisai Co., Ltd. (JP) 2002-08-14 EP disclosed
US-5792781-A EFFECTIVE AGAINST DERMATOMYCOSIS/VISCEROMYCOSIS CAUSED BY FUNGI, I.E., CANDIDA ALBICANS EISAI CO., LTD. (JP) 1998-08-11 US disclosed
US-5789429-A FUNGICIDE EISAI CO., LTD. (JP) 1998-08-04 US disclosed
US-5648372-A TRIAZOLES EISAI CO., LTD. (JP) 1997-07-15 US disclosed
EP-0667346-A2 Azole antifungal agents, process for the preparation there of and intermediates Eisai Co., Ltd. (JP) 1995-08-16 EP disclosed