SCHEMBL6630671

SCHEMBL6630671

NC(=O)c1ccc(Sc2ccccc2C(N)=O)cc1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT1 Q96EB6 3/20 0.77
PARP1 P09874 2/20 0.47
TDP1 Q9NUW8 2/20 0.47
MAPT P10636 2/20 0.47
TSHR P16473 2/20 0.47
HSD17B10 Q99714 2/20 0.47
CYP2C19 P33261 2/20 0.47
POLB P06746 1/20 0.47
CYP3A4 P08684 1/20 0.47
RECQL P46063 1/20 0.47
BLM P54132 1/20 0.47
PMP22 Q01453 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
BCL2L1 Q07817 1/20 0.46
ALDH1A1 P00352 3/20 0.43
KDM4E B2RXH2 2/20 0.43
HPGD P15428 3/20 0.42
PLA2G10 O15496 1/20 0.42
PLA2G2A P14555 1/20 0.42
GSTP1 P09211 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6630704 0.88 SIRT1 (0.70) SIRT1TDP1MAPTTSHRHSD17B10
SCHEMBL1030659 0.87 SIRT1 (1.00) SIRT1TDP1MAPTTSHRHSD17B10
SCHEMBL6627708 0.86 SIRT1 (0.77) SIRT1PARP1MAPTTSHRHSD17B10
SCHEMBL6630665 0.86 SIRT1 (0.77) SIRT1PARP1TDP1MAPTTSHR
SCHEMBL23018582 0.84 SIRT1 (0.55) SIRT1TDP1MAPTL3MBTL1BCL2L1
SCHEMBL11334883 0.84 SIRT1 (0.74) SIRT1MAPTPOLBBLML3MBTL1
SCHEMBL3077375 0.82 SIRT1 (0.77) SIRT1PARP1TDP1MAPTTSHR
SCHEMBL6632571 0.81 SIRT1 (0.70) SIRT1PARP1TDP1MAPTTSHR
SCHEMBL6129059 0.81 SIRT1 (0.50) SIRT1PARP1TDP1MAPTTSHR
SCHEMBL7695938 0.81 SIRT1 (0.74) SIRT1PARP1MAPTTSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1480977-A2 SUBSTITUTED ARYL COMPOUNDS FOR TREATMENT OF DISEASE PHARMACIA & UPJOHN COMPANY (US) 2004-12-01 EP claimed
WO-2003070728-A2 AZABICYCLO-SUBSTITUTED BENZOYLAMIDES AND THIOAMIDES FOR TREATMENT OF CNS-RELATED DISORDERS PHARMACIA & UPJOHN COMPANY (US) 2003-08-28 WO claimed