SCHEMBL6632172

SCHEMBL6632172

CC(C)[Si](O[C@@H](CS(=O)(=O)Cc1ccccc1)C(=O)NCCCC(=O)c1nc2ccccc2o1)(C(C)C)C(C)C

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DAGLA Q9Y4D2 11/20 0.47
FAAH O00519 6/20 0.47
CES1 P23141 3/20 0.47
XDH P47989 3/20 0.37
ALDH1A1 P00352 1/20 0.36
MTNR1A P48039 1/20 0.35
MTNR1B P49286 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6062697 0.87 DAGLA (0.47) DAGLAFAAHCES1XDHALDH1A1
SCHEMBL6061613 0.85 DAGLA (0.51) DAGLAFAAHCES1ALDH1A1
SCHEMBL6630749 0.84 DAGLA (0.53) DAGLAFAAHCES1XDHALDH1A1
SCHEMBL6063287 0.82 CTSS (0.46)
SCHEMBL6063280 0.82 CTSS (0.46)
SCHEMBL6062834 0.82 DAGLA (0.56) DAGLAFAAHCES1ALDH1A1
SCHEMBL6062952 0.82 DAGLA (0.52) DAGLAFAAHCES1XDHALDH1A1
SCHEMBL6631047 0.80 DAGLA (0.52) DAGLAFAAHCES1XDHALDH1A1
SCHEMBL6061646 0.80 DAGLA (0.48) DAGLAFAAHCES1ALDH1A1
SCHEMBL6061821 0.78 DAGLA (0.51) DAGLAFAAHCES1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1397340-A2 CHEMICAL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS AS CATHEPSIN S INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2004-03-17 EP claimed
WO-2002098850-A2 CHEMICAL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS AS CATHEPSIN S INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2002-12-12 WO claimed
EP-1397340-A2 CHEMICAL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS AS CATHEPSIN S INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2004-03-17 EP disclosed
WO-2002098850-A2 CHEMICAL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS AS CATHEPSIN S INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2002-12-12 WO disclosed