SCHEMBL6062697

SCHEMBL6062697

COCO[C@@H](CS(=O)(=O)Cc1ccccc1)C(=O)NCCCC(=O)c1nc2ccccc2o1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DAGLA Q9Y4D2 10/20 0.47
FAAH O00519 5/20 0.47
CES1 P23141 2/20 0.47
XDH P47989 2/20 0.37
ALDH1A1 P00352 1/20 0.36
RAB9A P51151 2/20 0.35
KDM4E B2RXH2 1/20 0.35
GLO1 Q04760 1/20 0.35
CTSS P25774 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6061613 0.88 DAGLA (0.51) DAGLAFAAHCES1ALDH1A1
SCHEMBL6632172 0.87 DAGLA (0.47) DAGLAFAAHCES1XDHALDH1A1
SCHEMBL6630749 0.84 DAGLA (0.53) DAGLAFAAHCES1XDHALDH1A1
SCHEMBL6062695 0.82 CTSS (0.47) CTSS
SCHEMBL6701293 0.82 CTSS (0.47) CTSS
SCHEMBL6062834 0.82 DAGLA (0.56) DAGLAFAAHCES1ALDH1A1
SCHEMBL6062952 0.80 DAGLA (0.52) DAGLAFAAHCES1XDHALDH1A1
SCHEMBL6631047 0.80 DAGLA (0.52) DAGLAFAAHCES1XDHALDH1A1
SCHEMBL6061646 0.80 DAGLA (0.48) DAGLAFAAHCES1ALDH1A1
SCHEMBL6062702 0.79 DAGLA (0.43) DAGLAFAAHCES1XDHRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1694357-A1 USE OF CATHEPSIN S INHIBITORS FOR TREATING AN IMMUNE RESPONSE CAUSED BY ADMINISTRATION OF A SMALL MOLECULE THERAPEUTIC OR BIOLOGIC AXYS PHARMACEUTICALS, INC. (US) 2006-08-30 EP disclosed
WO-2005058348-A1 USE OF CATHEPSIN S INHIBITORS FOR TREATING AN IMMUNE RESPONSE CAUSED BY ADMINISTRATION OF A SMALL MOLECULE THERAPEUTIC OR BIOLOGIC AXYS PHARMACEUTICALS, INC. (US) 2005-06-30 WO disclosed