SCHEMBL6633729

SCHEMBL6633729

Cc1ccc(S(=O)(=O)N2CCC[C@@H]2C(=O)N[C@@H](Cc2ccc(OC(=O)ON3CCN(OC(=O)Oc4ccc(C[C@H](NC(=O)[C@H]5CCCN5S(=O)(=O)c5ccc(C)cc5)C(=O)OC(C)C)cc4)CC3)cc2)C(=O)OC(C)C)cc1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 3/20 0.52
ITGB1 P05556 4/20 0.48
ITGB7 P26010 1/20 0.48
ITGA5 P08648 2/20 0.45
KMT2A Q03164 1/20 0.44
GAA P10253 1/20 0.44
HPGD P15428 1/20 0.44
FKBP1A P62942 2/20 0.44
ALDH1A1 P00352 1/20 0.44
MAPT P10636 1/20 0.43
HCRTR1 O43613 3/20 0.43
HCRTR2 O43614 3/20 0.43
MAPK1 P28482 2/20 0.43
TSHR P16473 1/20 0.43
CYP3A4 P08684 1/20 0.43
KCNQ1 P51787 1/20 0.43
RAB9A P51151 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6631919 0.90 ITGA4 (0.52) ITGA4ITGB1ITGB7ITGA5GAA
SCHEMBL3855551 0.89 ITGA4 (0.54) ITGA4ITGB1ITGB7ITGA5KMT2A
SCHEMBL3851005 0.88 ITGA4 (0.53) ITGA4ITGB1ITGB7ITGA5KMT2A
SCHEMBL3859212 0.86 ITGA4 (0.53) ITGA4ITGB1ITGB7ITGA5KMT2A
SCHEMBL5175369 0.86 ITGA4 (0.51) ITGA4ITGB1ITGB7ITGA5KMT2A
SCHEMBL7066750 0.86 FKBP1A (0.58) ITGA4ITGB1ITGA5GAAHPGD
SCHEMBL6708385 0.85 KMT2A (0.56) ITGA4ITGB1ITGA5KMT2AALDH1A1
SCHEMBL3849111 0.85 ITGA4 (0.51) ITGA4ITGB1ITGB7ITGA5KMT2A
SCHEMBL3853413 0.85 ITGA4 (0.51) ITGA4ITGB1ITGB7ITGA5KMT2A
SCHEMBL3850548 0.85 ITGA4 (0.50) ITGA4ITGB1ITGB7ITGA5KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1000051-B1 CARBAMYLOXY COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARM INC (US) 2004-05-19 EP claimed