SCHEMBL6633749

SCHEMBL6633749

Cn1c(COc2ccc(C(=N)N)cc2)nc2cc(NS(=O)(=O)CC3CCCCC3)ccc21

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
F2 P00734 13/20 0.51
F10 P00742 7/20 0.46
HDAC6 Q9UBN7 1/20 0.44
PRSS1 P07477 1/20 0.43
PRSS2 P07478 1/20 0.43
PRSS3 P35030 1/20 0.43
ALDH1A1 P00352 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8027015 0.87 F2 (0.65) F2F10PRSS1PRSS2PRSS3
SCHEMBL8026562 0.86 F2 (0.67) F2F10PRSS1PRSS2PRSS3
SCHEMBL6638105 0.86 F2 (0.57) F2F10PRSS1PRSS2PRSS3
SCHEMBL6635646 0.86 PPARG (0.43) F2HDAC6ALDH1A1
Hydrochloric Acid SCHEMBL8028460 0.86 F2 (0.66) F2F10PRSS1PRSS2PRSS3
SCHEMBL6640816 0.75 F2 (0.61) F2F10HDAC6PRSS1PRSS2
SCHEMBL8027045 0.74 F2 (0.45) F2ALDH1A1
SCHEMBL6633895 0.73 F2 (0.58) F2F10HDAC6PRSS1PRSS2
SCHEMBL8029893 0.72 F2 (0.46) F2
SCHEMBL6635980 0.72 SMN1; SMN2 (0.42) F2F10HDAC6PRSS1PRSS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1100795-B1 DISUBSTITUTED BICYCLIC HETEROCYCLES HAVING, IN PARTICULAR, A THROMBIN INHIBITIVE EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2004-06-09 EP disclosed
US-6121308-A INDOLE AND BENZIMIDAZOLE ANTITHROMBOTIC COMPOUNDS, SUCH AS 1-METHYL-2-(N-(4-AMIDINOPHENYL)-AMINOMETHYL)-5-(N-(HYDROXYCARBONYLMETHYL) -QUINOLINE-8-SULPHONYLAMINO)-INDOLE BOEHRINGER INGELHEIM KG (DE) 2000-09-19 US disclosed