SCHEMBL6635646

SCHEMBL6635646

Cn1c(COc2ccc(C#N)cc2)nc2cc(NS(=O)(=O)CC3CCCCC3)ccc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 1/20 0.43
LMNA P02545 4/20 0.41
ALDH1A1 P00352 2/20 0.41
HTT P42858 2/20 0.41
MEN1 O00255 1/20 0.41
HPGD P15428 1/20 0.41
KMT2A Q03164 1/20 0.41
USP2 O75604 1/20 0.40
F2 P00734 1/20 0.40
PKM P14618 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
TP53 P04637 1/20 0.40
THRB P10828 1/20 0.40
ALOX12 P18054 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
PAX8 Q06710 3/20 0.40
NPC1 O15118 1/20 0.40
POLB P06746 1/20 0.40
AURKA O14965 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8027045 0.88 F2 (0.45) LMNAALDH1A1HTTUSP2F2
SCHEMBL8029893 0.87 F2 (0.46) LMNAUSP2F2PKMSMN1; SMN2
SCHEMBL6635980 0.87 SMN1; SMN2 (0.42) LMNAALDH1A1HTTKMT2AUSP2
SCHEMBL6633749 0.86 F2 (0.51) ALDH1A1F2HDAC6
SCHEMBL6635652 0.77 PPARG (0.43) PPARGF2HDAC6NPC1AURKA
SCHEMBL6636883 0.72 SMN1; SMN2 (0.56) PPARGLMNAALDH1A1HTTHPGD
Hydrochloric Acid SCHEMBL8027015 0.72 F2 (0.65) F2NPC1
SCHEMBL8026562 0.71 F2 (0.67) F2
SCHEMBL6638105 0.71 F2 (0.57) F2
SCHEMBL6638614 0.71 F2 (0.43) PPARGLMNAALDH1A1HTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1100795-B1 DISUBSTITUTED BICYCLIC HETEROCYCLES HAVING, IN PARTICULAR, A THROMBIN INHIBITIVE EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2004-06-09 EP disclosed
US-6121308-A INDOLE AND BENZIMIDAZOLE ANTITHROMBOTIC COMPOUNDS, SUCH AS 1-METHYL-2-(N-(4-AMIDINOPHENYL)-AMINOMETHYL)-5-(N-(HYDROXYCARBONYLMETHYL) -QUINOLINE-8-SULPHONYLAMINO)-INDOLE BOEHRINGER INGELHEIM KG (DE) 2000-09-19 US disclosed