SCHEMBL6638545

SCHEMBL6638545

NC1Cn2cccc2Sc2ccccc21

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 1/20 0.42
DRD3 P35462 2/20 0.32
LMNA P02545 1/20 0.32
TP53 P04637 1/20 0.32
CYP2D6 P10635 1/20 0.32
TSHR P16473 1/20 0.32
CHRM2 P08172 1/20 0.32
HTR1A P08908 1/20 0.32
ADRA2A P08913 1/20 0.32
CHRM1 P11229 1/20 0.32
DRD1 P21728 1/20 0.32
TBXA2R P21731 1/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
ADRA1A P35348 1/20 0.32
OPRM1 P35372 1/20 0.32
KCNH2 Q12809 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32
DRD2 P14416 1/20 0.31
HTR2A P28223 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7495913 0.81 SLC6A3 (0.42) SLC6A3DRD3LMNATP53CYP2D6
SCHEMBL7494831 0.81 SLC6A3 (0.42) SLC6A3DRD3LMNATP53CYP2D6
SCHEMBL7494352 0.74 SLC6A3 (0.74) SLC6A3TP53CYP2D6TSHRDRD2
SCHEMBL7544150 0.66 SLC6A3 (0.61) SLC6A3TP53CYP2D6TSHRDRD2
SCHEMBL7494600 0.66 SLC6A3 (0.44) SLC6A3
SCHEMBL7495367 0.66 SLC6A3 (0.44) SLC6A3DRD3ADRA2ADRD1DRD2
SCHEMBL9693133 0.63 HTR2A (0.45) TP53CYP2D6TSHRHTR1ADRD2
SCHEMBL6779110 0.63 ANPEP (0.36) TP53CYP2D6HTR2A
SCHEMBL88255 0.62 HTR2A (0.46) SLC6A3DRD3LMNATP53CYP2D6
SCHEMBL8144693 0.61 HTR2A (0.41) SLC6A3DRD1SLC6A2SLC6A4HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1305318-B1 PROCESS FOR THE PREPARATION OF 9-AMINO SUBSTITUTED 9,10-DIHYDROPYRROLO [2,1-B] [1,3]BENZOTHIAZEPINES SIGMA TAU IND FARMACEUTI (IT) 2004-03-17 EP disclosed
EP-1305318-A1 PROCESS FOR THE PREPARATION OF 9-AMINO SUBSTITUTED 9,10-DIHYDROPYRROLO 2,1-B] 1,3]BENZOTIAZEPINES Sigma-Tau Industrie Farmaceutiche Riunite S.p.A. (IT) 2003-05-02 EP disclosed