SCHEMBL6638641

SCHEMBL6638641

c1ccc(CNCCc2ncc[nH]2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 2/20 0.57
GAA P10253 1/20 0.53
MAPT P10636 1/20 0.53
HRH4 Q9H3N8 1/20 0.51
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
TERT O14746 1/20 0.50
CYP2D6 P10635 1/20 0.48
TSHR P16473 1/20 0.48
LMNA P02545 1/20 0.47
GLA P06280 1/20 0.47
BLM P54132 1/20 0.47
PMP22 Q01453 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
SIGMAR1 Q99720 3/20 0.46
MAOA P21397 1/20 0.46
BCHE P06276 1/20 0.45
MPO P05164 1/20 0.45
PDCD1LG2 Q9BQ51 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9658713 0.91 TAAR1 (0.54) TAAR1GAAMAPTHRH4MEN1
SCHEMBL2475485 0.85 TAAR1 (0.62) TAAR1GAAMAPTMEN1KMT2A
SCHEMBL4775864 0.83 TERT (0.59) TAAR1TERTPDCD1LG2CD274
SCHEMBL12807572 0.80 TERT (0.66) TAAR1TERTPDCD1LG2CD274
SCHEMBL570036 0.79 TAAR1 (0.69) TAAR1TERTCYP2D6TSHRLMNA
Hydrochloric Acid SCHEMBL1846181 0.78 TAAR1 (0.67) TAAR1TERTCYP2D6TSHRLMNA
SCHEMBL9666999 0.77 TAAR1 (0.70) TAAR1GAAMAPTMEN1KMT2A
SCHEMBL15121693 0.76 TAAR1 (0.65) TAAR1TERTCYP2D6TSHRLMNA
SCHEMBL8958092 0.76 TAAR1 (0.65) TAAR1TERTCYP2D6TSHRLMNA
SCHEMBL9370948 0.76 POLB (0.49) TAAR1HRH4TERTCYP2D6LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1322309-A4 HIGH AFFINITY SMALL MOLECULE C5A RECEPTOR MODULATORS NEUROGEN CORP (US) 2004-10-13 EP disclosed
EP-1322309-A2 HIGH AFFINITY SMALL MOLECULE C5A RECEPTOR MODULATORS Neurogen Corporation (US) 2003-07-02 EP disclosed
WO-2002049993-A2 HIGH AFFINITY SMALL MOLECULE C5A RECEPTOR MODULATORS NEUROGEN CORPORATION (US) 2002-06-27 WO disclosed