SCHEMBL6640168

SCHEMBL6640168

COc1cc2c(C)nccc2cc1Cl

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNF P01375 4/20 0.47
SRC P12931 1/20 0.46
CGAS Q8N884 1/20 0.44
CYP3A4 P08684 3/20 0.42
PDE10A Q9Y233 3/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
ACHE P22303 3/20 0.42
USP2 O75604 2/20 0.42
ALDH1A1 P00352 2/20 0.42
LMNA P02545 2/20 0.42
CYP1A2 P05177 2/20 0.42
CYP2D6 P10635 2/20 0.42
CYP2C9 P11712 2/20 0.42
MAPK1 P28482 2/20 0.42
CYP2C19 P33261 2/20 0.42
PDE3B Q13370 2/20 0.42
PDE3A Q14432 2/20 0.42
HIF1A Q16665 2/20 0.42
PDE2A O00408 1/20 0.42
ABCC4 O15439 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3974591 0.86 CYP3A4 (0.54) TNFCYP3A4PDE10ASMN1; SMN2ACHE
SCHEMBL30458203 0.86 CYP3A4 (0.54) TNFCYP3A4PDE10ASMN1; SMN2ACHE
SCHEMBL17278085 0.83 MAPT (0.45) TNFCYP3A4PDE10ASMN1; SMN2ACHE
SCHEMBL16431495 0.80 APAF1 (0.48) TNFCYP3A4PDE10ASMN1; SMN2ACHE
SCHEMBL1536597 0.78 TNF (0.48) TNFSRCCGASCYP3A4PDE10A
SCHEMBL16431829 0.77 APAF1 (0.48) TNFCYP3A4PDE10ASMN1; SMN2ACHE
SCHEMBL14538274 0.77 TRPA1 (0.54) TNFCYP3A4PDE10ASMN1; SMN2ACHE
SCHEMBL31589356 0.74 TNF (0.57) TNFCYP3A4PDE10ASMN1; SMN2ACHE
SCHEMBL5358941 0.74 TNF (0.57) TNFCYP3A4PDE10ASMN1; SMN2ACHE
SCHEMBL8271696 0.73 TRPA1 (0.51) TNFSRCCYP3A4PDE10ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0867436-B1 N-aryl-piperidine derivatives and their use as 5-HT1B receptor ligands SERVIER LAB (FR) 2004-06-09 EP disclosed
US-5965575-A N-aryl piperidine compounds as 5HT1B antagonists ADIR ET COMPAGNIE (FR) 1999-10-12 US disclosed
EP-0867436-A1 N-aryl-piperidine derivatives and their use as 5-HT1B receptor ligands ADIR ET COMPAGNIE (FR) 1998-09-30 EP disclosed