SCHEMBL6640344

SCHEMBL6640344

N=C(N)c1ccc(CC(=O)N2CCc3ccc(N(CC(=O)O)S(=O)(=O)c4cccc5cccnc45)cc3C2)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F2 P00734 6/20 0.60
ALDH1A1 P00352 3/20 0.41
HTT P42858 2/20 0.40
KDM4E B2RXH2 1/20 0.40
HPGD P15428 1/20 0.40
HSD17B10 Q99714 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
POLB P06746 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
ALOX15 P16050 1/20 0.39
TSHR P16473 1/20 0.39
MAPK1 P28482 1/20 0.39
TP53 P04637 2/20 0.38
STS P08842 2/20 0.38
ESR1 P03372 1/20 0.38
OXTR P30559 1/20 0.37
AVPR1A P37288 1/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.36
ITGB3 P05106 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6635794 0.90 F2 (0.51) F2ALDH1A1HTTKDM4EHPGD
Hydrochloric Acid SCHEMBL6636092 0.81 F2 (0.56) F2
SCHEMBL6976662 0.80 F2 (0.60) F2ALDH1A1HTTPOLBNPSR1
SCHEMBL6635719 0.78 ALDH1A1 (0.40) F2ALDH1A1HTTKDM4EHPGD
Hydrochloric Acid SCHEMBL7361185 0.76 F2 (0.66) F2ALDH1A1HPGDLMNAMAPT
SCHEMBL6635405 0.75 F2 (0.78) F2ALDH1A1HPGDSMN1; SMN2MAPT
Hydrochloric Acid SCHEMBL8016304 0.75 F2 (0.76) F2ALDH1A1HPGDMAPT
SCHEMBL8027337 0.75 F2 (1.00) F2
SCHEMBL7424644 0.75 F2 (0.83) F2
SCHEMBL8124847 0.75 F2 (0.69) F2ALDH1A1HTTHPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1100795-B1 DISUBSTITUTED BICYCLIC HETEROCYCLES HAVING, IN PARTICULAR, A THROMBIN INHIBITIVE EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2004-06-09 EP disclosed
US-6121308-A INDOLE AND BENZIMIDAZOLE ANTITHROMBOTIC COMPOUNDS, SUCH AS 1-METHYL-2-(N-(4-AMIDINOPHENYL)-AMINOMETHYL)-5-(N-(HYDROXYCARBONYLMETHYL) -QUINOLINE-8-SULPHONYLAMINO)-INDOLE BOEHRINGER INGELHEIM KG (DE) 2000-09-19 US disclosed