SCHEMBL6640489

SCHEMBL6640489

Nc1cc(Cl)nc(SCc2c(F)cccc2F)n1

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
RAB9A P51151 5/20 0.51
NPC1 O15118 3/20 0.51
PKM P14618 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
SMN1; SMN2 Q16637 5/20 0.46
TOP2A P11388 1/20 0.45
KDM4E B2RXH2 1/20 0.44
TP53 P04637 1/20 0.44
MPO P05164 2/20 0.40
LMNA P02545 1/20 0.40
DCK P27707 2/20 0.40
NFKB1 P19838 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6641351 0.85 SMN1; SMN2 (0.56) MEN1KMT2ARAB9ANPC1PKM
SCHEMBL490008 0.85 NPC1 (0.48) MEN1KMT2ARAB9ANPC1SMN1; SMN2
SCHEMBL1520900 0.84 MPO (0.54) MEN1KMT2ARAB9ANPC1SMN1; SMN2
SCHEMBL6639107 0.82 RAB9A (0.51) MEN1KMT2ARAB9ANPC1PKM
SCHEMBL8136755 0.80 RAB9A (0.49) MEN1KMT2ARAB9ANPC1PKM
SCHEMBL1520700 0.80 RAB9A (0.81) MEN1KMT2ARAB9ANPC1SMN1; SMN2
SCHEMBL490086 0.79 MPO (0.48) MEN1KMT2ARAB9ANPC1PKM
SCHEMBL490002 0.78 MEN1 (0.61) MEN1KMT2ARAB9ANPC1SMN1; SMN2
SCHEMBL489860 0.77 RAB9A (0.78) MEN1KMT2ARAB9ANPC1SMN1; SMN2
SCHEMBL490003 0.77 MEN1 (0.59) MEN1KMT2ARAB9ANPC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1449835-A2 Alpha-substituted pyrimidine-thioalkyl and alkylether compounds PHARMACIA & UPJOHN COMPANY (US) 2004-08-25 EP disclosed
EP-1247804-A1 Pyrimidine-thioalkyl and alkylether compounds PHARMACIA & UPJOHN COMPANY (US) 2002-10-09 EP disclosed
US-6043248-A VIRICIDES FOR TREATING AN INDIVIDUAL INFECTED WITH THE HUMAN IMMUNODEFICIENCY VIRUS PHARMACIA & UPJOHN COMPANY (US) 2000-03-28 US disclosed
US-5981537-A USEFUL IN THE TREATMENT OF INDIVIDUALS WHO ARE HIV POSITIVE PHARMACIA & UPJOHN COMPANY (US) 1999-11-09 US disclosed
EP-0824524-A1 ALPHA-SUBSTITUTED PYRIMIDINE-THIOALKYL AND ALKYLETHER COMPOUNDS AS INHIBITORS OF VIRAL REVERSE TRANSCRIPTASE PHARMACIA & UPJOHN COMPANY (US) 1998-02-25 EP disclosed
EP-0728130-A1 PYRIMIDINE-THIOALKYL AND ALKYLETHER COMPOUNDS PHARMACIA & UPJOHN COMPANY (US) 1996-08-28 EP disclosed
WO-1995013267-A1 PYRIMIDINE-THIOALKYL AND ALKYLETHER COMPOUNDS THE UPJOHN COMPANY (US) 1995-05-18 WO disclosed