SCHEMBL6640934

SCHEMBL6640934

CCc1ccnc([C@@H](C)O)c1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.50
NOS1 P29475 1/20 0.50
NOS2 P35228 1/20 0.50
TRPA1 O75762 1/20 0.36
SMYD3 Q9H7B4 1/20 0.35
RIOK2 Q9BVS4 1/20 0.35
SORD Q00796 1/20 0.35
CTSA P10619 2/20 0.34
PKM P14618 1/20 0.34
AKR1C3 P42330 1/20 0.33
AKR1C2 P52895 1/20 0.33
RECQL P46063 1/20 0.33
ADRB2 P07550 1/20 0.33
KCNA5 P22460 1/20 0.33
CYP1A2 P05177 1/20 0.33
POLB P06746 1/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6636590 1.00 NOS3 (0.50) NOS3NOS1NOS2TRPA1SMYD3
SCHEMBL2737265 0.84 NOS3 (0.53) NOS3NOS1NOS2TRPA1SMYD3
SCHEMBL6638502 0.81 HRH3 (0.39) PKMRECQLPOLBMEN1KMT2A
SCHEMBL20889614 0.81 NOS3 (0.55) NOS3NOS1NOS2SMYD3CTSA
SCHEMBL17778607 0.78 NOS3 (0.52) NOS3NOS1NOS2TRPA1SMYD3
SCHEMBL21185561 0.78 NOS3 (0.47) NOS3NOS1NOS2TRPA1SMYD3
SCHEMBL18945314 0.78 NOS3 (0.47) NOS3NOS1NOS2TRPA1SMYD3
SCHEMBL27028346 0.74 KMT2A (0.47) NOS1NOS2AKR1C3AKR1C2MEN1
SCHEMBL27845901 0.74 ADRB2 (0.31) SORDADRB2KCNA5
SCHEMBL27028354 0.74 KMT2A (0.47) NOS1NOS2AKR1C3AKR1C2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1535958-A Alpha-substituted pyrimidine. thioalkyl and alkyl ether compound �������Ŷ���Լ��������˾ 2004-10-13 CN disclosed
EP-0824524-B1 ALPHA-SUBSTITUTED PYRIMIDINE-THIOALKYL AND ALKYLETHER COMPOUNDS AS INHIBITORS OF VIRAL REVERSE TRANSCRIPTASE UPJOHN CO (US) 2004-09-08 EP disclosed
EP-1449835-A2 Alpha-substituted pyrimidine-thioalkyl and alkylether compounds PHARMACIA & UPJOHN COMPANY (US) 2004-08-25 EP disclosed
CN-1152022-C Alpha-substituted pyrimidine-thioalkyl and alkylether compounds �������Ŷ���Լ��������˾ 2004-06-02 CN disclosed
US-6043248-A VIRICIDES FOR TREATING AN INDIVIDUAL INFECTED WITH THE HUMAN IMMUNODEFICIENCY VIRUS PHARMACIA & UPJOHN COMPANY (US) 2000-03-28 US disclosed
CN-1183773-A Alpha-substituted pyrimidine-thioalkyl and alkylether compounds UPJOHN CO (US) 1998-06-03 CN disclosed
WO-1996035678-A1 ALPHA-SUBSTITUTED PYRIMIDINE-THIOALKYL AND ALKYLETHER COMPOUNDS AS INHIBITORS OF VIRAL REVERSE TRANSCRIPTASE PHARMACIA & UPJOHN COMPANY (US) 1996-11-14 WO disclosed